Target Details
| UniProt AC | O60341 |
|---|---|
| Gene Symbol | KDM1A |
| Protein Name | Lysine-specific histone demethylase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01593 (Amino_oxidase) PF04433 (SWIRM) |
Summary
- Multi-target molecules 721
- Clinical molecules 0
- Avg pChEMBL 7.55
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (721)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LZDNSUQSFKCUBO
|
7.2 | IC50 | 2 | — | |
VQXSHYNCIQFRBL
|
7.2 | IC50 | 3 | — | |
XLPPGAPESQIJTN
|
7.2 | IC50 | 2 | — | |
HEOKXBMRYSEMPZ
|
7.2 | IC50 | 2 | — | |
LCJHHBITOMGPDB
|
7.2 | IC50 | 3 | — | |
TVQYDGRYNLMFHN
|
7.2 | IC50 | 2 | — | |
CRFTYPZVLZZIHU
|
7.2 | IC50 | 2 | — | |
HJSROIWRJOQVCL
|
7.2 | IC50 | 2 | — | |
IYOQBCSTSLISOI
|
7.2 | IC50 | 2 | — | |
RUFLTUCAFVGHGI
|
7.2 | IC50 | 2 | — | |
YSMJYMKVLSNDRL
|
7.2 | IC50 | 2 | — | |
ZVVDKVJEGXSFFZ
|
7.2 | IC50 | 2 | — | |
PNLZPOBONAJYFY
|
7.2 | IC50 | 2 | — | |
ZRCDNYZZNYQDNU
|
7.2 | IC50 | 2 | — | |
MDWANQHRPJNECZ
|
7.2 | IC50 | 2 | — | |
UYUHYANMQFXLMI
|
7.2 | IC50 | 2 | — | |
WVVHNLMQBRBRGZ
|
7.2 | IC50 | 2 | — | |
DQVINXBYDSVKBR
|
7.2 | IC50 | 2 | — | |
OOUPHCVQCFQHLO
|
7.2 | IC50 | 2 | — | |
QAZSEXHFQQZAIT
|
7.2 | IC50 | 2 | — | |
ASCMSQYWEMJWFA
|
7.2 | IC50 | 2 | — | |
BLXYCLXIDWUQPD
|
7.1 | IC50 | 2 | — | |
SSKPQHGCUVMGAQ
|
7.1 | IC50 | 2 | — | |
PEINCKFKYMDPOM
|
7.1 | IC50 | 3 | — | |
ZPIKKAOXWOJZTG
|
7.1 | IC50 | 2 | — | |
ATCXSBVZCGQDCJ
|
7.1 | IC50 | 2 | — | |
DHKMEXBVLDKGIA
|
7.1 | IC50 | 2 | — | |
NXKYPBDDPFDALC
|
7.1 | IC50 | 3 | — | |
NTYPTMOHHKHCRO
|
7.1 | IC50 | 2 | — | |
PSRVWCBORZIYDW
|
7.1 | Ki | 2 | — | |
QXRFQNQVZQAPGV
|
7.1 | IC50 | 2 | — | |
RZPJSFNGGGHGEC
|
7.1 | IC50 | 2 | — | |
YGALSGSYVHMATA
|
7.1 | IC50 | 2 | — | |
KZVAKSHUKOLEJK
|
7.1 | IC50 | 2 | — | |
SMXGFVZOSHQEFC
|
7.1 | IC50 | 2 | — | |
WGTZIEXXJINMNT
|
7.1 | IC50 | 2 | — | |
ZFDITTSJGFSWMG
|
7.1 | Kd | 2 | — | |
GJXFBKDQIXYBIK
|
7.1 | IC50 | 2 | — | |
HFOCUYHVEWLYRP
|
7.1 | IC50 | 2 | — | |
HZDYKFBUGRBRMH
|
7.1 | IC50 | 2 | — | |
BINXOHRETRQOCW
|
7.1 | IC50 | 2 | — | |
CLMKFAVBRRFUGX
|
7.1 | Kd | 2 | — | |
YJZRGYKZHFUFLQ
|
7.1 | IC50 | 3 | — | |
ZPIXRPPZFQFTJS
|
7.1 | IC50 | 2 | — | |
SNNSGPYMBKEIBR
|
7.1 | IC50 | 2 | — | |
UFKPGWMKQUSRPU
|
7.1 | IC50 | 2 | — | |
AAPZDXBWJBCGRD
|
7.0 | IC50 | 2 | — | |
BINXOHRETRQOCW
|
7.0 | IC50 | 2 | — | |
IZUMRIVGTVNLDD
|
7.0 | IC50 | 2 | — | |
LWVYBAUVCPWKSM
|
7.0 | IC50 | 2 | — |