Target Details
| UniProt AC | O60341 |
|---|---|
| Gene Symbol | KDM1A |
| Protein Name | Lysine-specific histone demethylase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01593 (Amino_oxidase) PF04433 (SWIRM) |
Summary
- Multi-target molecules 721
- Clinical molecules 0
- Avg pChEMBL 7.55
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (721)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RHYDLZPXYPVUIP
|
7.4 | IC50 | 2 | — | |
UJVNULKJXOXHLR
|
7.4 | IC50 | 3 | — | |
BUTMZXYDLXMRED
|
7.3 | Ki | 2 | — | |
FFQGGLINEZDCSL
|
7.3 | IC50 | 2 | — | |
WGTSRMDFUQLHJX
|
7.3 | IC50 | 2 | — | |
ZWMGUAYLVFCVEL
|
7.3 | IC50 | 2 | — | |
PTHMQEMZNPDKLO
|
7.3 | IC50 | 2 | — | |
QRPWGONVHSCJTL
|
7.3 | IC50 | 2 | — | |
QZNGFWQWWSECMG
|
7.3 | IC50 | 2 | — | |
JAOMJGNNLHDGIP
|
7.3 | IC50 | 2 | — | |
PJRFPYJEXUAIAO
|
7.3 | IC50 | 2 | — | |
TVPSDFDZPXEOIQ
|
7.3 | IC50 | 2 | — | |
YCAWTMXHBSTPQD
|
7.3 | IC50 | 2 | — | |
BINXOHRETRQOCW
|
7.3 | IC50 | 2 | — | |
GJRDYRHJJPYKSV
|
7.3 | IC50 | 3 | — | |
PEIUICYITJBEGE
|
7.3 | IC50 | 2 | — | |
LSTXXVDRMNZSAI
|
7.3 | IC50 | 3 | — | |
YIPPIWJAJVYULJ
|
7.3 | IC50 | 2 | — | |
ALHBJBCQLJZYON
|
7.3 | IC50 | 2 | — | |
CBHJAQSSOXSUFD
|
7.3 | IC50 | 3 | — | |
CQCWLDROOQGZAS
|
7.3 | Ki | 3 | — | |
HDVDLEPVLVTECB
|
7.3 | IC50 | 2 | — | |
HJWZUPRHNBJKHE
|
7.3 | Ki | 2 | — | |
IHSXBANMVVFXGY
|
7.3 | Ki | 2 | — | |
JRNQFIYVQYTRHZ
|
7.3 | Ki | 2 | — | |
KXDUCUANSPMTGM
|
7.3 | Ki | 3 | — | |
NUABRMQYIQQHPM
|
7.3 | Ki | 2 | — | |
PMGVDYFOLLPRPE
|
7.3 | Ki | 2 | — | |
SNZBTOXJQFMTHW
|
7.3 | Ki | 2 | — | |
SOYHGUPORKZZJR
|
7.3 | Ki | 2 | — | |
XLZPYWFUNBTRGV
|
7.3 | IC50 | 3 | — | |
ZWIYKBPLUJMBJN
|
7.3 | Ki | 2 | — | |
IFINDMLSYQDICS
|
7.3 | IC50 | 2 | — | |
NSWDBAURHGVFRJ
|
7.3 | IC50 | 3 | — | |
TVQYDGRYNLMFHN
|
7.3 | IC50 | 2 | — | |
ALHBJBCQLJZYON
|
7.3 | IC50 | 2 | — | |
BINXOHRETRQOCW
|
7.3 | IC50 | 2 | — | |
JEGXEQPWCZLZQF
|
7.3 | IC50 | 2 | — | |
NKOGAETYSHVEAL
|
7.3 | IC50 | 2 | — | |
MCZRLRYBKZHKLE
|
7.3 | IC50 | 2 | — | |
VLTIYMVMEIUCSB
|
7.3 | IC50 | 3 | — | |
KSNYGZADPGAMKR
|
7.2 | IC50 | 2 | — | |
FPEFNMXJYVYZLS
|
7.2 | IC50 | 2 | — | |
LONLDQWPQKYQPD
|
7.2 | IC50 | 2 | — | |
NUHULANAKMSLMG
|
7.2 | IC50 | 2 | — | |
SBZNZJNYVPWQPU
|
7.2 | Ki | 2 | — | |
WIQHXHNUMWQTDT
|
7.2 | IC50 | 2 | — | |
BHRMTBMFKWLVQR
|
7.2 | IC50 | 2 | — | |
FICFTOMKYYZSEL
|
7.2 | IC50 | 4 | — | |
JEZAGOJTCWQABS
|
7.2 | IC50 | 2 | — |