Target Details
| UniProt AC | O60341 |
|---|---|
| Gene Symbol | KDM1A |
| Protein Name | Lysine-specific histone demethylase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01593 (Amino_oxidase) PF04433 (SWIRM) |
Summary
- Multi-target molecules 721
- Clinical molecules 0
- Avg pChEMBL 7.55
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (721)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CGFMLQROEREMOV
|
7.7 | IC50 | 2 | — | |
FFYGOYSNGFPHEN
|
7.7 | IC50 | 3 | — | |
IQVDLEXWAPYWDT
|
7.7 | IC50 | 2 | — | |
NZNSESWVOLCQQL
|
7.7 | IC50 | 2 | — | |
UMQFLXROKIABBY
|
7.7 | IC50 | 2 | — | |
OPGHKNVSNFWTCM
|
7.7 | IC50 | 3 | — | |
SJXSJRJEKZWPGE
|
7.7 | IC50 | 3 | — | |
BAPMAOYONKAQPM
|
7.7 | IC50 | 3 | — | |
FFYGOYSNGFPHEN
|
7.7 | IC50 | 2 | — | |
GWSJKJBRTAYFIO
|
7.7 | IC50 | 2 | — | |
GWSJKJBRTAYFIO
|
7.7 | IC50 | 2 | — | |
HQRYNOVKRKLADI
|
7.7 | IC50 | 2 | — | |
JZVXHLNIORJHPD
|
7.7 | IC50 | 2 | — | |
JZVXHLNIORJHPD
|
7.7 | IC50 | 2 | — | |
MIKODFRFXKEMPU
|
7.7 | IC50 | 2 | — | |
NALIOKLWLFSTCV
|
7.7 | IC50 | 2 | — | |
NALIOKLWLFSTCV
|
7.7 | IC50 | 2 | — | |
OAZVHMYGOGQYLZ
|
7.7 | IC50 | 2 | — | |
QMOFHXLCMXQBLM
|
7.7 | IC50 | 2 | — | |
DDEBLIXHOWDGMM
|
7.7 | IC50 | 4 | — | |
BWTYCKXFSJVJTA
|
7.6 | IC50 | 2 | — | |
FXKFQJGJMSTPFG
|
7.6 | IC50 | 2 | — | |
VORPELBVCZFEBS
|
7.6 | IC50 | 2 | — | |
VORPELBVCZFEBS
|
7.6 | IC50 | 2 | — | |
DESMZSTXYFPMPK
|
7.6 | IC50 | 2 | — | |
JELFJCHCBUKLFJ
|
7.6 | IC50 | 2 | — | |
MULCJXMWOPKAQH
|
7.6 | IC50 | 2 | — | |
NVCODPCMEFURSY
|
7.6 | IC50 | 2 | — | |
SAAIALQMXUSENU
|
7.6 | IC50 | 2 | — | |
CBZDXOREIVGUGU
|
7.6 | IC50 | 3 | — | |
ICFNLJYZHKCEMV
|
7.6 | IC50 | 2 | — | |
BGYXCRFJBFJHGH
|
7.6 | IC50 | 2 | — | |
IINYVTZTXIVCOR
|
7.6 | IC50 | 2 | — | |
ONDFAHAVDKQBCV
|
7.6 | IC50 | 2 | — | |
FFYGOYSNGFPHEN
|
7.6 | IC50 | 2 | — | |
YMMYPJZLMRASOA
|
7.6 | IC50 | 2 | — | |
IJWYHMIMXOCAJF
|
7.6 | IC50 | 2 | — | |
LWCLBPGSSWFOQV
|
7.6 | IC50 | 2 | — | |
QTRSQEGGLVSWCR
|
7.6 | IC50 | 2 | — | |
VUUUJQSTZWEXHY
|
7.6 | IC50 | 2 | — | |
YZUHPMZFIGGUPF
|
7.6 | IC50 | 2 | — | |
BQOHMXILIJCNFY
|
7.5 | IC50 | 2 | — | |
HFFNZRXCDSLUQO
|
7.5 | IC50 | 2 | — | |
IKJFIPIKSOKVSV
|
7.5 | IC50 | 3 | — | |
AJYWAQNMQLIZQD
|
7.5 | IC50 | 2 | — | |
AWLSYOBVZBVGNU
|
7.5 | IC50 | 2 | — | |
BBPDDMYSLCWVDE
|
7.5 | IC50 | 2 | — | |
DCFLYLYZNLKCEM
|
7.5 | IC50 | 2 | — | |
KEXPXBUNMVXDSV
|
7.5 | IC50 | 2 | — | |
PBSVFESALQWDIE
|
7.5 | IC50 | 3 | — |