Target Details
| UniProt AC | O60341 |
|---|---|
| Gene Symbol | KDM1A |
| Protein Name | Lysine-specific histone demethylase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01593 (Amino_oxidase) PF04433 (SWIRM) |
Summary
- Multi-target molecules 721
- Clinical molecules 0
- Avg pChEMBL 7.55
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (721)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZPIXRPPZFQFTJS
|
8.1 | IC50 | 2 | — | |
BEPWDOKDBUCNJP
|
8.1 | IC50 | 3 | — | |
KMEAOGUGZPSHRG
|
8.1 | IC50 | 3 | — | |
SOFOPIVHMPQVDO
|
8.1 | IC50 | 3 | — | |
QGGLLHNPYXLEQQ
|
8.1 | IC50 | 2 | — | |
SUJXSOKWACSDJM
|
8.0 | IC50 | 3 | — | |
WWTVNHCOQIGYHP
|
8.0 | IC50 | 3 | — | |
PKTXMHFXTNPAEM
|
8.0 | IC50 | 2 | — | |
PYDFVFWGGDZAOA
|
8.0 | IC50 | 2 | — | |
IJRPMLXEUJPAFM
|
8.0 | IC50 | 2 | — | |
JKRNUDVNHUULRR
|
8.0 | IC50 | 2 | — | |
JVYBRGTXJDGJBA
|
8.0 | IC50 | 3 | — | |
DTMDFPAJMNVMBI
|
8.0 | IC50 | 3 | — | |
UOHSMFGBWNRISH
|
8.0 | IC50 | 3 | — | |
UMCMUHXVQOVKIH
|
8.0 | IC50 | 2 | — | |
UMCMUHXVQOVKIH
|
8.0 | IC50 | 2 | — | |
HGQXBRHZRCCGGT
|
7.9 | IC50 | 2 | — | |
HOJXWPCFCRGBLU
|
7.9 | IC50 | 2 | — | |
VPWONGMLZUGDBA
|
7.9 | IC50 | 2 | — | |
FFYGOYSNGFPHEN
|
7.9 | IC50 | 2 | — | |
XNCFADKPSKGXFW
|
7.9 | IC50 | 2 | — | |
LBJKNBQOIJJEFH
|
7.9 | IC50 | 2 | — | |
SHRXGXDMIAZWHE
|
7.9 | IC50 | 2 | — | |
VVGBYNYCWGLRCF
|
7.9 | IC50 | 3 | — | |
KFBVBYZQLWHGSI
|
7.9 | IC50 | 2 | — | |
YAMSXCOVJUUMCT
|
7.8 | IC50 | 2 | — | |
ZHNSGNCXGXHASO
|
7.8 | IC50 | 3 | — | |
AHHNXKYEHPZBNR
|
7.8 | IC50 | 3 | — | |
KUHOELRKSJUYCN
|
7.8 | IC50 | 2 | — | |
KUHOELRKSJUYCN
|
7.8 | IC50 | 2 | — | |
BPHDDXANELGDOF
|
7.8 | IC50 | 2 | — | |
KVHQXEXKAHCVTD
|
7.8 | IC50 | 2 | — | |
OZGYPGKEBOFBFZ
|
7.8 | IC50 | 2 | — | |
VVDRSVLMDANHHP
|
7.8 | IC50 | 3 | — | |
XQOVXGUKFBOUSX
|
7.8 | IC50 | 2 | — | |
VKNZCFMDYLENSQ
|
7.8 | IC50 | 3 | — | |
ALHBJBCQLJZYON
|
7.8 | IC50 | 3 | — | |
ALHBJBCQLJZYON
|
7.7 | IC50 | 4 | — | |
OAZVHMYGOGQYLZ
|
7.7 | IC50 | 2 | — | |
WDKFNHQULODPEI
|
7.7 | IC50 | 2 | — | |
FODIXKGYNUVLOV
|
7.7 | IC50 | 3 | — | |
OGIMVYIRQGYCPV
|
7.7 | IC50 | 2 | — | |
GVFVFSPQLVQDNV
|
7.7 | IC50 | 2 | — | |
VPZPSTHUSDFUKN
|
7.7 | IC50 | 2 | — | |
VPZPSTHUSDFUKN
|
7.7 | IC50 | 2 | — | |
XNOVADVADHFJFS
|
7.7 | IC50 | 2 | — | |
NSOIWQGZHDVJTN
|
7.7 | IC50 | 2 | — | |
NTRMVYTYDOLCRU
|
7.7 | IC50 | 2 | — | |
BNWKPONIDAHKBK
|
7.7 | IC50 | 2 | — | |
BNWKPONIDAHKBK
|
7.7 | IC50 | 2 | — |