Target Details
| UniProt AC | O60341 |
|---|---|
| Gene Symbol | KDM1A |
| Protein Name | Lysine-specific histone demethylase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01593 (Amino_oxidase) PF04433 (SWIRM) |
Summary
- Multi-target molecules 721
- Clinical molecules 0
- Avg pChEMBL 7.55
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (721)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FOHNOCWNMWVRNN
|
8.5 | IC50 | 2 | — | |
PSKKUNLHYZLZMX
|
8.5 | IC50 | 2 | — | |
CDTNICJXZZUXTQ
|
8.5 | IC50 | 2 | — | |
OBWIFFLIJZFZAI
|
8.5 | IC50 | 3 | — | |
QBWSSNPGKOQCHT
|
8.5 | IC50 | 3 | — | |
QTWMTAMDRGVNEQ
|
8.5 | IC50 | 2 | — | |
VVSVLJROTRDBRW
|
8.5 | IC50 | 2 | — | |
GLBCFKBDVDVHJN
|
8.4 | IC50 | 3 | — | |
MYGPMSRCVMTNSR
|
8.4 | IC50 | 2 | — | |
VUPIIHSYRDZCSU
|
8.4 | IC50 | 2 | — | |
HACUHRDPZRXYSI
|
8.4 | IC50 | 2 | — | |
KWBPNWHUYTYXFB
|
8.4 | IC50 | 2 | — | |
KWBPNWHUYTYXFB
|
8.4 | IC50 | 2 | — | |
VBTIXCLUYQDMRA
|
8.4 | IC50 | 2 | — | |
APWSULSJYLPFPF
|
8.4 | IC50 | 3 | — | |
GWADQWPCNFDVIN
|
8.4 | IC50 | 3 | — | |
OLWIXPHBDXNLPR
|
8.4 | IC50 | 3 | — | |
BWJWLFNSMWKGSY
|
8.4 | IC50 | 2 | — | |
IRTGGRPCQKEPED
|
8.4 | IC50 | 3 | — | |
XZGHKNIRCDWQDK
|
8.4 | IC50 | 3 | — | |
RHFCADKDRKOCST
|
8.4 | IC50 | 3 | — | |
AELCINSCMGFISI
|
8.3 | IC50 | 4 | — | |
DAKWITGIEKEPRZ
|
8.3 | IC50 | 2 | — | |
QYCZNZQEXYMDOH
|
8.3 | IC50 | 3 | — | |
SGFIWDBZENQUHG
|
8.3 | IC50 | 2 | — | |
FPWRGPARLXITJF
|
8.3 | IC50 | 2 | — | |
HACUHRDPZRXYSI
|
8.3 | IC50 | 2 | — | |
QGGLLHNPYXLEQQ
|
8.3 | IC50 | 2 | — | |
RSEQCKDWYUJYAC
|
8.3 | IC50 | 2 | — | |
CTRYUUQZYMUPNG
|
8.3 | IC50 | 2 | — | |
HACUHRDPZRXYSI
|
8.2 | IC50 | 3 | — | |
HOJXWPCFCRGBLU
|
8.2 | IC50 | 2 | — | |
HQQZDZUCNFOPJH
|
8.2 | IC50 | 2 | — | |
HQQZDZUCNFOPJH
|
8.2 | IC50 | 2 | — | |
PCYSURNBQUNXFM
|
8.2 | IC50 | 2 | — | |
PCYSURNBQUNXFM
|
8.2 | IC50 | 2 | — | |
JJOOKDGBBREJDT
|
8.2 | IC50 | 3 | — | |
VUAJJNFTKHBMLV
|
8.2 | IC50 | 3 | — | |
XTIUXFVWQDSKHY
|
8.2 | IC50 | 2 | — | |
VUKSNWXXGOMEJT
|
8.2 | IC50 | 2 | — | |
ZNPKDAJYJOBTSM
|
8.1 | IC50 | 2 | — | |
ZZLBFEKJJDCLHD
|
8.1 | IC50 | 2 | — | |
DZODKSZEJNSJMA
|
8.1 | IC50 | 2 | — | |
SQSNNQXVJVEDMY
|
8.1 | IC50 | 2 | — | |
CTNAJMVWCJOHQE
|
8.1 | IC50 | 3 | — | |
HOJXWPCFCRGBLU
|
8.1 | IC50 | 2 | — | |
KHQVACSLVNHFEZ
|
8.1 | IC50 | 2 | — | |
TXZHNZXQIYCIQP
|
8.1 | IC50 | 2 | — | |
BVNIBOGSMAIXSI
|
8.1 | IC50 | 2 | — | |
IRZLLRSBKUBRSE
|
8.1 | IC50 | 3 | — |