Target Details
| UniProt AC | O60341 |
|---|---|
| Gene Symbol | KDM1A |
| Protein Name | Lysine-specific histone demethylase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01593 (Amino_oxidase) PF04433 (SWIRM) |
Summary
- Multi-target molecules 721
- Clinical molecules 0
- Avg pChEMBL 7.55
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (721)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NUPNPRUYOLMBRH
|
8.9 | IC50 | 3 | — | |
MZIBJUYAKXQIDU
|
8.9 | IC50 | 3 | — | |
AZTHAJKEPBKWIZ
|
8.9 | IC50 | 3 | — | |
NHZDNAPDBMZQAH
|
8.9 | IC50 | 3 | — | |
UTMQDIUPSJGZGI
|
8.9 | IC50 | 3 | — | |
WAKHYXWQFQTCFM
|
8.9 | IC50 | 3 | — | |
RIIJKPSGJSZLGY
|
8.9 | IC50 | 3 | — | |
PBSMCYGDPUAIEK
|
8.8 | IC50 | 3 | — | |
SPCWBSDMJZUPMU
|
8.8 | IC50 | 2 | — | |
ZHKPPPCBDXKUGR
|
8.8 | IC50 | 3 | — | |
DUNDWPGZRFAQLI
|
8.8 | IC50 | 2 | — | |
QJLHXFWIJAZQSJ
|
8.8 | IC50 | 2 | — | |
WUPAKHUDFAJWNH
|
8.8 | IC50 | 3 | — | |
DFMAVPKQECRLCK
|
8.8 | IC50 | 3 | — | |
OMPCGMQBVCKNFU
|
8.8 | IC50 | 2 | — | |
DLBZBSURVFVXPO
|
8.8 | IC50 | 3 | — | |
KOPQPXVNOUMQLP
|
8.8 | IC50 | 3 | — | |
HULMGLKQHMUCSC
|
8.8 | IC50 | 3 | — | |
URQHUOKPZBICBP
|
8.8 | IC50 | 3 | — | |
KPIQXEHVUNOBJE
|
8.8 | IC50 | 2 | — | |
OKIKDKJGIUQYLE
|
8.8 | IC50 | 3 | — | |
BKTQCQFRBAQVAT
|
8.8 | IC50 | 3 | — | |
PPVYNJSPWYEUQX
|
8.7 | IC50 | 2 | — | |
XLRFJYPISMPMNU
|
8.7 | IC50 | 3 | — | |
XXNBWGMYBZLSFN
|
8.7 | IC50 | 3 | — | |
ZKHWWYQXKUMLOY
|
8.7 | IC50 | 3 | — | |
LYXITNHLBNAMBP
|
8.7 | IC50 | 2 | — | |
MVVNZEUTFJHGQC
|
8.7 | IC50 | 3 | — | |
MXSOGWIOQMYTHA
|
8.7 | IC50 | 3 | — | |
FSSPLVOEHOXMJK
|
8.7 | IC50 | 2 | — | |
DZNWAGBPQLJDFO
|
8.7 | IC50 | 3 | — | |
IZRBKNQECMLOJZ
|
8.7 | IC50 | 2 | — | |
IZRBKNQECMLOJZ
|
8.7 | IC50 | 2 | — | |
BJVPULRQOIWJGY
|
8.7 | IC50 | 3 | — | |
SAFYJSRSFACVJV
|
8.7 | IC50 | 2 | — | |
WOSQQPZAYPSCNQ
|
8.7 | IC50 | 3 | — | |
XMZOVQCTCRRWJP
|
8.7 | IC50 | 3 | — | |
DTOMUHCXYBDCDT
|
8.6 | IC50 | 3 | — | |
ASQRMWZGHICKTE
|
8.6 | IC50 | 2 | — | |
XUXJOXZUGGOEEU
|
8.6 | IC50 | 2 | — | |
XZFIOYRHNYMHHE
|
8.6 | IC50 | 2 | — | |
KUBWSUSDCQEXTO
|
8.6 | IC50 | 2 | — | |
VNMDZVXDBWIRLR
|
8.6 | IC50 | 3 | — | |
NKXZTUSRLWODTJ
|
8.6 | IC50 | 3 | — | |
VKLQJRUWNXXNPX
|
8.6 | IC50 | 3 | — | |
VMVFOYPCQRCISD
|
8.6 | IC50 | 3 | — | |
FXEYLIGKDAKHFG
|
8.6 | IC50 | 3 | — | |
JGRDDJKBSGFALE
|
8.6 | IC50 | 3 | — | |
QZNGFWQWWSECMG
|
8.5 | IC50 | 2 | — | |
CXVZFKHTYDMSLH
|
8.5 | IC50 | 2 | — |