Target Details
| UniProt AC | O60341 |
|---|---|
| Gene Symbol | KDM1A |
| Protein Name | Lysine-specific histone demethylase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01593 (Amino_oxidase) PF04433 (SWIRM) |
Summary
- Multi-target molecules 721
- Clinical molecules 0
- Avg pChEMBL 7.55
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (721)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PMNMXEZSVZEZSS
|
9.3 | IC50 | 3 | — | |
SCHADMXEZDXOLS
|
9.2 | IC50 | 3 | — | |
XOQLULSVIJENMN
|
9.2 | IC50 | 3 | — | |
XYSKEBYDGKOLCW
|
9.2 | IC50 | 3 | — | |
SGOVVPUUSBJRBP
|
9.2 | IC50 | 3 | — | |
WSNOUIZBNPNLIJ
|
9.2 | IC50 | 2 | — | |
YKNCRTIRHJDVKM
|
9.2 | IC50 | 3 | — | |
KAVQRNLEDUQHCY
|
9.2 | IC50 | 3 | — | |
PSEAJFICJHBQJD
|
9.2 | IC50 | 3 | — | |
YRFNCDCBEHRSQD
|
9.2 | IC50 | 3 | — | |
BTGHQTJZAWUBCC
|
9.2 | IC50 | 2 | — | |
IWLAILJDCGZCOX
|
9.2 | IC50 | 2 | — | |
LTLDVPDLHXMPQM
|
9.2 | IC50 | 2 | — | |
MTJZAYKBPCGSNH
|
9.2 | IC50 | 3 | — | |
PFYIRZUNGVGORR
|
9.2 | IC50 | 3 | — | |
NLOAXXMZUZFADG
|
9.1 | IC50 | 3 | — | |
IJIUCUSMQWXDFW
|
9.1 | IC50 | 3 | — | |
WFXUCMWHLZFYTJ
|
9.1 | IC50 | 3 | — | |
WRARGVGMPKUUTH
|
9.1 | IC50 | 3 | — | |
MGEGEFWEBBYEDQ
|
9.1 | IC50 | 3 | — | |
IZCZUGBFAJALOV
|
9.1 | IC50 | 3 | — | |
LYNZHNLVMDLVOS
|
9.1 | IC50 | 2 | — | |
SMTWFEJFHSIPKD
|
9.1 | IC50 | 2 | — | |
GYHURJUXWPDQFH
|
9.1 | IC50 | 3 | — | |
SICZWEWEDUOACO
|
9.1 | IC50 | 2 | — | |
XHLRZJKTRQULGZ
|
9.1 | IC50 | 2 | — | |
HGYQCPBGWSBYEB
|
9.0 | IC50 | 2 | — | |
VHIYYWZBVPLQNW
|
9.0 | IC50 | 2 | — | |
CTDCXRSZNSKWMK
|
9.0 | IC50 | 3 | — | |
IRQFXBUIHHIUTI
|
9.0 | IC50 | 2 | — | |
JPKHNASOORDOLS
|
9.0 | IC50 | 3 | — | |
KFAWNIPYOUVGFI
|
9.0 | IC50 | 3 | — | |
SBMQWRXZUUXWSP
|
9.0 | IC50 | 2 | — | |
PUPPIJVQIIPCRT
|
9.0 | IC50 | 3 | — | |
HDQOUBINEKYXPX
|
9.0 | IC50 | 3 | — | |
XBILHKJVQHPCOM
|
9.0 | IC50 | 3 | — | |
FKERNWUYZXDWFM
|
9.0 | IC50 | 3 | — | |
NBGAFGGNFMNQTJ
|
9.0 | IC50 | 3 | — | |
YZUBULKCVYIFGL
|
9.0 | IC50 | 3 | — | |
IHCLVMILZHMPOZ
|
9.0 | IC50 | 2 | — | |
YAFAYFUCWHRMBW
|
9.0 | IC50 | 3 | — | |
DLLWVCLKELQMAF
|
8.9 | IC50 | 3 | — | |
DWEYHCDIQVLBOP
|
8.9 | IC50 | 3 | — | |
GKENUJVDMFBCDM
|
8.9 | IC50 | 3 | — | |
WUIBJHPAWAMRFO
|
8.9 | IC50 | 3 | — | |
HPKIXQIFZBOYMA
|
8.9 | IC50 | 3 | — | |
BMJAWOGCGUEVGD
|
8.9 | IC50 | 3 | — | |
WTGMUNCNXTUDSC
|
8.9 | IC50 | 3 | — | |
NAEVJSGKGLNYFG
|
8.9 | IC50 | 3 | — | |
XSGVWOISEZRQQQ
|
8.9 | IC50 | 3 | — |