Target Details
| UniProt AC | O60341 |
|---|---|
| Gene Symbol | KDM1A |
| Protein Name | Lysine-specific histone demethylase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01593 (Amino_oxidase) PF04433 (SWIRM) |
Summary
- Multi-target molecules 721
- Clinical molecules 0
- Avg pChEMBL 7.55
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (721)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MUNCZXCTDJVHER
|
7.0 | IC50 | 3 | — | |
YSHCPCIXRXSLEV
|
7.0 | IC50 | 2 | — | |
ITHUGPBMQIDROK
|
7.0 | IC50 | 3 | — | |
BINXOHRETRQOCW
|
7.0 | IC50 | 2 | — | |
FUXLXWZVYUFWPI
|
7.0 | IC50 | 2 | — | |
JWUGFZWTKOOIHE
|
7.0 | IC50 | 2 | — | |
UXBZYLRHNRJDCG
|
7.0 | IC50 | 2 | — | |
CAVFCZTWZCRFBW
|
7.0 | IC50 | 2 | — | |
WUZBFLILHSCABF
|
7.0 | IC50 | 2 | — | |
FOGVZOPDYOPZAB
|
7.0 | Kd | 2 | — | |
ZFEJPJCYTLSKFD
|
7.0 | IC50 | 2 | — | |
AHOWVATWFHRVFS
|
7.0 | IC50 | 3 | — | |
FNFVTNNWNCYKMO
|
7.0 | IC50 | 2 | — | |
KHMZBPOHQQODIO
|
7.0 | IC50 | 2 | — | |
LTQDYSVREOECNH
|
7.0 | IC50 | 2 | — | |
NDNVIFQCNJINSJ
|
7.0 | IC50 | 2 | — | |
RIILCHKMPVLDAX
|
7.0 | IC50 | 2 | — | |
SASCNLRSTSEASB
|
7.0 | IC50 | 2 | — | |
YMULIXZFUBPIGR
|
7.0 | IC50 | 2 | — | |
YTHOTLCZYQVYSA
|
7.0 | IC50 | 2 | — | |
ONJAKTJSPHBUNM
|
7.0 | IC50 | 2 | — | |
ONJAKTJSPHBUNM
|
7.0 | IC50 | 2 | — | |
KCVSNHFBVOJMIT
|
7.0 | IC50 | 2 | — | |
RREBWWQLLSXJPH
|
7.0 | IC50 | 2 | — | |
BSMLOLVDLSYQAE
|
7.0 | IC50 | 2 | — | |
FPEFNMXJYVYZLS
|
7.0 | IC50 | 2 | — | |
IZYGIQRTVUJNEH
|
7.0 | IC50 | 2 | — | |
SKAXHFHMJFPVDU
|
7.0 | Kd | 2 | — | |
SOBRGCVHDJATAI
|
7.0 | IC50 | 2 | — | |
BAHNEQQCLXPUQN
|
7.0 | IC50 | 2 | — | |
CCBZNXUXMQHMLT
|
7.0 | IC50 | 2 | — | |
KNLMZFKJTDDDQH
|
7.0 | Kd | 3 | — | |
NRRVBNCEYIEHLS
|
7.0 | IC50 | 2 | — | |
OTVUAMDWWYQCKJ
|
7.0 | IC50 | 2 | — | |
UAQFERXHHSHKOB
|
7.0 | Kd | 2 | — | |
YKDCWZQOYSBNAE
|
7.0 | Kd | 2 | — | |
NNYGHETYMLXJTD
|
7.0 | Kd | 2 | — | |
NDNVIFQCNJINSJ
|
6.9 | IC50 | 2 | — | |
XXSQTUAKUSHIBV
|
6.9 | Kd | 2 | — | |
PDOPAKBSLLNWSO
|
6.9 | IC50 | 2 | — | |
COYFSGVVDODYNC
|
6.9 | IC50 | 2 | — | |
JSXHMKTUCJTVHQ
|
6.9 | IC50 | 2 | — | |
KTGNPKLCQXMRCO
|
6.9 | IC50 | 2 | — | |
OCNOGEHYMVMKEE
|
6.9 | IC50 | 2 | — | |
PIZBQXXOLNPHSO
|
6.9 | Kd | 2 | — | |
QLTFOHFSLUPAAG
|
6.9 | IC50 | 2 | — | |
UBPRBNRVPWGYDA
|
6.9 | Kd | 2 | — | |
VQDWAJLSYJGIDH
|
6.9 | IC50 | 2 | — | |
CIDSRGYSMPCJCV
|
6.9 | IC50 | 2 | — | |
CWUHUYVZKXLJGU
|
6.9 | IC50 | 2 | — |