Target Details
| UniProt AC | O60341 |
|---|---|
| Gene Symbol | KDM1A |
| Protein Name | Lysine-specific histone demethylase 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01593 (Amino_oxidase) PF04433 (SWIRM) |
Summary
- Multi-target molecules 721
- Clinical molecules 0
- Avg pChEMBL 7.55
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (721)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BPAPNYGEUHCUDM
|
10.7 | IC50 | 2 | — | |
REMZJIYFJDROFR
|
10.5 | IC50 | 2 | — | |
PLNPDHQHVIPIPU
|
10.4 | IC50 | 3 | — | |
KCUDVBBQWGIKPW
|
10.3 | IC50 | 3 | — | |
AISFXQFMHKDBSQ
|
10.2 | IC50 | 3 | — | |
DOBGCSDZOYQKSP
|
10.1 | IC50 | 3 | — | |
VTDHBGCLTJFGHR
|
10.1 | IC50 | 2 | — | |
WSEGJZJJHCUQPA
|
10.1 | IC50 | 3 | — | |
GKGLKZKLMWNIJS
|
10.0 | IC50 | 3 | — | |
PNQKDRVYVUAGJA
|
10.0 | IC50 | 3 | — | |
GKPWROMXYMULQP
|
10.0 | IC50 | 2 | — | |
PHFRWNDMBDKWAC
|
9.9 | IC50 | 2 | — | |
UOMQFBUEOBYYHG
|
9.9 | IC50 | 3 | — | |
UATQZZVNCXYTBX
|
9.8 | IC50 | 2 | — | |
WXMJOABDWLLAKI
|
9.8 | IC50 | 3 | — | |
IXAGWRIVLLNVFN
|
9.8 | IC50 | 3 | — | |
NHKPSJXKMXGDNU
|
9.7 | IC50 | 2 | — | |
RQZLGLMWTFNKEP
|
9.7 | IC50 | 2 | — | |
KJDDLVZUCZDGQS
|
9.7 | IC50 | 3 | — | |
LJUBVENCCNSBMK
|
9.6 | IC50 | 3 | — | |
XPNGHMNQWWEIDK
|
9.6 | IC50 | 3 | — | |
GEPUWBAMAOGGDT
|
9.6 | IC50 | 2 | — | |
FZMHPVGYWUFSIQ
|
9.5 | IC50 | 3 | — | |
RHVKPGJHMLOYTQ
|
9.5 | IC50 | 3 | — | |
RVRYILXECYBQQE
|
9.5 | IC50 | 2 | — | |
FWPYWZSRFRWCAZ
|
9.5 | IC50 | 3 | — | |
NYJMZHMGSDOBCG
|
9.5 | IC50 | 3 | — | |
ZEUYYAFLPVPYDQ
|
9.5 | IC50 | 3 | — | |
ZSDBZVOFOUNISV
|
9.5 | IC50 | 2 | — | |
XGKMCBYRFZHMBO
|
9.4 | IC50 | 3 | — | |
MNHUURYMAORLLV
|
9.4 | IC50 | 3 | — | |
ZCCPLJOKGAACRT
|
9.4 | Kd | 599 | — | |
PSOZICNDRAQYQP
|
9.4 | IC50 | 2 | — | |
TZKAPLJIEQYVTG
|
9.4 | IC50 | 3 | — | |
FYOYFMLTMWNXAU
|
9.4 | IC50 | 3 | — | |
SDJFMUFEDIEHMY
|
9.4 | IC50 | 3 | — | |
YAHBPBSMUNEMKG
|
9.4 | IC50 | 3 | — | |
NOYMCCHFPVFENX
|
9.4 | IC50 | 2 | — | |
OUISIOJCZOYDGY
|
9.4 | IC50 | 2 | — | |
WVZBQUZVOYIGLK
|
9.4 | IC50 | 3 | — | |
BBTFQCLFEDJYSY
|
9.4 | IC50 | 3 | — | |
HNQVHLDWWXSADR
|
9.4 | IC50 | 3 | — | |
AIEQMVYBDDVIPP
|
9.3 | IC50 | 3 | — | |
YJMOPUOJIHUJII
|
9.3 | IC50 | 3 | — | |
XBBRLCXCBCZIOI
|
9.3 | IC50 | 2 | — | |
FGYOOZLOHGPAER
|
9.3 | IC50 | 3 | — | |
NFJKAIPDHURTLR
|
9.3 | IC50 | 2 | — | |
NSYRUCCRJGQMNS
|
9.3 | IC50 | 3 | — | |
MCHRWCJFZOKWSN
|
9.3 | IC50 | 3 | — | |
NYHGGWMGKMXOEH
|
9.3 | IC50 | 3 | — |