Target Details
| UniProt AC | O60307 |
|---|---|
| Gene Symbol | MAST3 |
| Protein Name | Microtubule-associated serine/threonine-protein kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08926 (DUF1908) PF17820 (PDZ_6) PF00069 (Pkinase) |
Summary
- Multi-target molecules 7
- Clinical molecules 0
- Avg pChEMBL 6.18
Associated Diseases (1)
Active Molecules (7)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YOOLXKXFWTXRHM
|
6.6 | IC50 | 2 | — | |
KLRKVNKANBJQPN
|
6.5 | IC50 | 3 | — | |
MFJOWCFANZXQBU
|
6.1 | IC50 | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
WRXMCDABCCZKSX
|
6.0 | IC50 | 2 | — |