Target Details
| UniProt AC | O60285 |
|---|---|
| Gene Symbol | NUAK1 |
| Protein Name | NUAK family SNF1-like kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 57
- Clinical molecules 11
- Avg pChEMBL 7.35
Active Molecules (57)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TVJRAGSLXXBXQQ
|
6.2 | IC50 | 2 | — | |
OYONTEXKYJZFHA
|
6.2 | Kd | 69 | Yes | |
YBYYWUUUGCNAHQ
|
6.2 | IC50 | 8 | — | |
SWIVJTVGOIXUKC
|
6.1 | IC50 | 9 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |