Target Details
| UniProt AC | O60285 |
|---|---|
| Gene Symbol | NUAK1 |
| Protein Name | NUAK family SNF1-like kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 57
- Clinical molecules 11
- Avg pChEMBL 7.35
Active Molecules (57)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
8.8 | IC50 | 408 | — | |
FCLPVPNWFDOVKL
|
8.8 | Ki | 11 | — | |
JLWGOAGEDWMEBT
|
8.7 | IC50 | 10 | — | |
JLWGOAGEDWMEBT
|
8.7 | IC50 | 10 | — | |
LZUYOYKXEXENTQ
|
8.5 | IC50 | 5 | — | |
OFIFLUFVENTCNZ
|
8.5 | IC50 | 11 | — | |
SBLCPBDVMUSESZ
|
8.4 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
8.4 | Kd | 289 | Yes | |
LYADGAGFYYXXIO
|
8.4 | IC50 | 82 | — | |
HKSZLNNOFSGOKW
|
8.4 | Kd | 213 | — | |
VAVXGGRQQJZYBL
|
8.3 | IC50 | 8 | — | |
XLFNLJYGUOLEJS
|
8.3 | IC50 | 26 | — | |
SDGJBAUIGHSMRI
|
8.3 | IC50 | 3 | — | |
PHENCDSAYZNXRO
|
8.2 | IC50 | 3 | — | |
MJSHVHLADKXCML
|
8.1 | IC50 | 11 | — | |
NOMBUNHXDWBICV
|
8.1 | Ki | 11 | — | |
WGWCRXQUBYJTRA
|
8.0 | Ki | 11 | — | |
OSVUGUHRKMMBSE
|
7.9 | Kd | 170 | — | |
QQWUGDVOUVUTOY
|
7.9 | Kd | 231 | Yes | |
NXSJMRCTGYTSTK
|
7.8 | Kd | 200 | — | |
QNABDSWBQJKBHK
|
7.8 | IC50 | 45 | — | |
UEFCSGDOOJJXTN
|
7.7 | IC50 | 46 | — | |
ITTRLTNMFYIYPA
|
7.6 | IC50 | 17 | — | |
LAJAFFLJAJMYLK
|
7.6 | IC50 | 17 | — | |
MFWHDFGMXHATNR
|
7.5 | IC50 | 3 | — | |
JOOXLOJCABQBSG
|
7.5 | Kd | 139 | — | |
BMGQWWVMWDBQGC
|
7.4 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
7.4 | Kd | 91 | Yes | |
RSFALMGMTQBFJZ
|
7.4 | Kd | 9 | — | |
AILRADAXUVEEIR
|
7.3 | IC50 | 75 | — | |
WINHZLLDWRZWRT
|
7.3 | Kd | 201 | Yes | |
DOTGPNHGTYJDEP
|
7.2 | IC50 | 8 | — | |
NHHQJBCNYHBUSI
|
7.1 | Kd | 220 | — | |
ZZSBPGIGIUFJRA
|
7.0 | Kd | 46 | — | |
CJQGLUJHMXCLQY
|
6.9 | IC50 | 11 | — | |
ZHOXAGNPCZTRBN
|
6.8 | Kd | 20 | — | |
XZXHXSATPCNXJR
|
6.8 | Kd | 165 | Yes | |
RDROKTFULACVDQ
|
6.8 | IC50 | 8 | — | |
FTIGOWUZQQHANO
|
6.8 | IC50 | 3 | — | |
KDKUVYLMPJIGKA
|
6.7 | Kd | 91 | Yes | |
GCIKSSRWRFVXBI
|
6.7 | Kd | 109 | Yes | |
NGFGTMFVWSDFPS
|
6.7 | IC50 | 32 | — | |
UKBGBACORPRCGG
|
6.6 | IC50 | 17 | — | |
PIQCTGMSNWUMAF
|
6.6 | Kd | 137 | Yes | |
OEZHSZIDGUKBRK
|
6.5 | IC50 | 10 | — | |
HVIGNZUDBVLTLU
|
6.4 | IC50 | 7 | — | |
KUQOZTZPJMJBMT
|
6.4 | IC50 | 3 | — | |
KGPGFQWBCSZGEL
|
6.4 | Kd | 59 | Yes | |
CTNPALGJUAXMMC
|
6.3 | Kd | 151 | — | |
KPUGXRVRDQQZRP
|
6.2 | IC50 | 2 | — |