Target Details
| UniProt AC | O60259 |
|---|---|
| Gene Symbol | KLK8 |
| Protein Name | Kallikrein-8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00089 (Trypsin) |
Summary
- Multi-target molecules 14
- Clinical molecules 0
- Avg pChEMBL 6.84
Active Molecules (14)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NWAGTUQRZPXSNY
|
8.2 | IC50 | 6 | — | |
NWAGTUQRZPXSNY
|
7.6 | IC50 | 5 | — | |
NWAGTUQRZPXSNY
|
7.5 | IC50 | 4 | — | |
QFJOOWSJASQPAX
|
7.0 | IC50 | 7 | — | |
IVGMDANEFALECQ
|
6.9 | IC50 | 5 | — | |
CSTAEACZUNFQMP
|
6.8 | IC50 | 3 | — | |
CTDHLROQTKJDLK
|
6.8 | IC50 | 4 | — | |
UHZDIMFNWHQJEY
|
6.7 | IC50 | 3 | — | |
LUNUFGFUBAQPEV
|
6.6 | IC50 | 4 | — | |
OCOZTJLWHRDAJG
|
6.6 | IC50 | 4 | — | |
OPVLRSNIYJHUNK
|
6.5 | IC50 | 4 | — | |
YENXZRUMZHNJKP
|
6.4 | IC50 | 4 | — | |
WYCVSPRVSFUVMA
|
6.1 | IC50 | 3 | — | |
ZDLCAMFQMDNCSU
|
6.1 | IC50 | 2 | — |