Target Details
| UniProt AC | O60218 |
|---|---|
| Gene Symbol | AKR1B10 |
| Protein Name | Aldo-keto reductase family 1 member B10 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00248 (Aldo_ket_red) |
Summary
- Multi-target molecules 39
- Clinical molecules 0
- Avg pChEMBL 7.66
KEGG Pathways (6)
Active Molecules (39)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IRTLXYIOFBGNOF
|
8.5 | IC50 | 5 | — | |
YNGXWVIJSUJZSG
|
8.5 | IC50 | 5 | — | |
QEQGIVVMPNNCOY
|
8.3 | IC50 | 2 | — | |
ANZFBALHOWVGKN
|
8.2 | IC50 | 2 | — | |
PTODCHFEJHFEOL
|
8.2 | IC50 | 2 | — | |
VFNPSKKBRLJDNM
|
8.2 | IC50 | 2 | — | |
LHPNUZXMXZJHCT
|
8.2 | IC50 | 2 | — | |
XMAOASZNRJCMLI
|
8.2 | IC50 | 2 | — | |
CWHACJJNROINNY
|
8.1 | IC50 | 2 | — | |
PTJHHAABQXVCFD
|
8.1 | IC50 | 2 | — | |
VHBFRXWQXCNSTM
|
8.1 | IC50 | 2 | — | |
HOXOCVYGMMQSGX
|
8.1 | IC50 | 2 | — | |
IAMAUDKQJHVKCU
|
8.1 | IC50 | 2 | — | |
YLLFDRHTELGUAX
|
8.1 | IC50 | 2 | — | |
RWVPKZVHNKOTQF
|
8.0 | IC50 | 2 | — | |
GFTAMXNPASWXKC
|
8.0 | IC50 | 2 | — | |
GWBRUFXAFPGUAJ
|
8.0 | IC50 | 2 | — | |
ZLRZNGZTDMERMQ
|
8.0 | IC50 | 2 | — | |
ZUNCLGAPQBIVCJ
|
8.0 | IC50 | 2 | — | |
FZFWFVUOKSKHOO
|
7.9 | IC50 | 2 | — | |
VDFQWTHPVPUSSE
|
7.9 | IC50 | 2 | — | |
YFEMXNMSQVETGA
|
7.9 | IC50 | 2 | — | |
VFTQMEMIHPBYLO
|
7.9 | IC50 | 2 | — | |
UILYKFFFBGSSBC
|
7.8 | IC50 | 2 | — | |
ZNJRNZXFJKLDOI
|
7.8 | IC50 | 2 | — | |
NQWSOKVRUVPYSN
|
7.7 | IC50 | 2 | — | |
ZUULNQQNTCHGJQ
|
7.7 | IC50 | 2 | — | |
XPJSDAVSTGFBKS
|
7.7 | IC50 | 2 | — | |
FLCMSIBUTPDBOT
|
7.5 | IC50 | 2 | — | |
LUBHDINQXIHVLS
|
7.3 | IC50 | 3 | — | |
PREBVFJICNPEKM
|
7.2 | IC50 | 2 | — | |
GUMNIDBFNHVRBD
|
7.2 | IC50 | 2 | — | |
MIJYXULNPSFWEK
|
7.0 | Ki | 8 | — | |
RGZZCZQQPNJCPO
|
6.9 | IC50 | 7 | — | |
BCSVCWVQNOXFGL
|
6.2 | IC50 | 3 | — | |
BMHZAHGTGIZZCT
|
6.1 | IC50 | 3 | — | |
BMHZAHGTGIZZCT
|
6.1 | IC50 | 3 | — | |
LPEPZBJOKDYZAD
|
6.1 | IC50 | 7 | — | |
WVDDMJTWFGHTGZ
|
6.0 | IC50 | 7 | — |