Target Details
| UniProt AC | O43781 |
|---|---|
| Gene Symbol | DYRK3 |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 301
- Clinical molecules 4
- Avg pChEMBL 6.64
Active Molecules (301)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FAIHBCXQSBIRIL
|
6.1 | Ki | 22 | — | |
HDEZJSLYUKYKAZ
|
6.1 | Ki | 6 | — | |
KAEULNCNLILYLK
|
6.1 | IC50 | 4 | — | |
RPGBQFNDFPEOON
|
6.1 | Ki | 22 | — | |
UYJNQQDJUOUFQJ
|
6.1 | Ki | 68 | — | |
VAMDLIMJLAPZGX
|
6.1 | Ki | 10 | — | |
YWTBGJGMTBHQTM
|
6.1 | Ki | 65 | — | |
BULHRWBHKAVJMT
|
6.1 | IC50 | 8 | — | |
NNPWUWSWEGWPMQ
|
6.1 | IC50 | 8 | — | |
VCCCOYOXNKTQFO
|
6.1 | IC50 | 9 | — | |
YMIDGKZVYFXIBW
|
6.1 | IC50 | 8 | — | |
USSKXRGFNVFHFF
|
6.1 | IC50 | 7 | — | |
BULHRWBHKAVJMT
|
6.1 | IC50 | 8 | — | |
GHQYHWMWJLSKRP
|
6.1 | IC50 | 9 | — | |
LZTDWHFXSWDVAG
|
6.1 | IC50 | 7 | — | |
OQGLPYHETIJRBX
|
6.1 | IC50 | 3 | — | |
OQGLPYHETIJRBX
|
6.1 | IC50 | 3 | — | |
URXJBXVGNBGIJA
|
6.1 | IC50 | 9 | — | |
MLGGUGPIWDHBAI
|
6.0 | Ki | 33 | — | |
RVSPPVBZRQFLQY
|
6.0 | IC50 | 6 | — | |
ZHTZVZJNJGCSJO
|
6.0 | IC50 | 7 | — | |
CEWIXDGUKGVYDQ
|
6.0 | IC50 | 7 | — | |
FTGAOPZDJRWUTG
|
6.0 | IC50 | 6 | — | |
HTNKXRHQVGPWRO
|
6.0 | IC50 | 3 | — | |
QGGNWMQODZFHNG
|
6.0 | IC50 | 4 | — | |
WREJZZXSNOJGIW
|
6.0 | IC50 | 8 | — | |
CTXSEYUOXKGIMM
|
6.0 | IC50 | 3 | — | |
UMYSGMXAOXMMGG
|
6.0 | IC50 | 7 | — | |
YELPLVUUDHOICI
|
6.0 | IC50 | 4 | — | |
ZQZULRTVXPNQNP
|
6.0 | IC50 | 4 | — | |
CSNGPDJYNPSXNA
|
6.0 | IC50 | 5 | — | |
MFLKPCAUPXBTPC
|
6.0 | IC50 | 6 | — | |
OAKDCYWBXLUPQD
|
6.0 | IC50 | 4 | — | |
PDJLHUHTIYCYTA
|
6.0 | IC50 | 4 | — | |
ACOQCSBMVFAWQV
|
6.0 | IC50 | 8 | — | |
AOBLBPWPSKBHSI
|
6.0 | Ki | 55 | — | |
BLTVBQXJFVRPFK
|
6.0 | Ki | 7 | — | |
DJUSDFVEBBYFFL
|
6.0 | Ki | 27 | — | |
FGLPGUCHBHILNS
|
6.0 | Ki | 10 | — | |
KJVWCDAPVMWKLJ
|
6.0 | Ki | 20 | — | |
MCCCQFAOMZMZKE
|
6.0 | Ki | 52 | — | |
NLUPJKQOKWBWFC
|
6.0 | Ki | 69 | — | |
PEXKNSGOEOREKM
|
6.0 | Ki | 13 | — | |
PSCJSWRVCKUMSL
|
6.0 | Ki | 35 | — | |
PSYVPXWWLKLHBA
|
6.0 | Ki | 2 | — | |
RAUYTJLQISREEJ
|
6.0 | Ki | 2 | — | |
VIJBEUTVNBPGIU
|
6.0 | Ki | 19 | — | |
WINHZLLDWRZWRT
|
6.0 | Ki | 66 | — | |
XCTYEZWILVGTGO
|
6.0 | IC50 | 9 | — | |
YHZQZEGQCKWCLP
|
6.0 | IC50 | 9 | — |