Target Details
| UniProt AC | O43781 |
|---|---|
| Gene Symbol | DYRK3 |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 301
- Clinical molecules 4
- Avg pChEMBL 6.64
Active Molecules (301)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MEKFXUFACKZUCV
|
6.3 | IC50 | 9 | — | |
WEQRXDXDFLBIDK
|
6.3 | IC50 | 8 | — | |
WFOMWAYINPJPDX
|
6.3 | IC50 | 9 | — | |
JBWDTSLHUJHODF
|
6.3 | IC50 | 8 | — | |
DCHAEDURAZJASA
|
6.2 | IC50 | 9 | — | |
DXVSNYWBRDTHFF
|
6.2 | IC50 | 7 | — | |
LXQXBEIFOYAXOP
|
6.2 | IC50 | 9 | — | |
YSBCFQVEEKUZSU
|
6.2 | IC50 | 7 | — | |
JXQZHHAAJMQJKU
|
6.2 | IC50 | 9 | — | |
QQCCFMCJVKPTMI
|
6.2 | IC50 | 4 | — | |
UXIAMCZUNQBRTJ
|
6.2 | IC50 | 4 | — | |
CUIDQTVRAWOMCM
|
6.2 | Ki | 7 | Yes | |
DXVSNYWBRDTHFF
|
6.2 | IC50 | 9 | — | |
FSWFKKQQSQHIRZ
|
6.2 | Ki | 10 | — | |
HHSVICUMCOBRPT
|
6.2 | Ki | 33 | — | |
IJNGXROUMFEKDB
|
6.2 | Ki | 39 | — | |
JOIUJUJSHIHBDT
|
6.2 | Ki | 18 | — | |
KCKXYZOBGBJZEG
|
6.2 | Ki | 36 | — | |
KXPWWMPXNUOYOH
|
6.2 | Ki | 24 | — | |
NWAUBAGBGOPJLF
|
6.2 | Ki | 51 | Yes | |
ODNOTLMFNVWFTJ
|
6.2 | Ki | 11 | — | |
OLVBAUVSICCWEJ
|
6.2 | Ki | 39 | — | |
VQPBIJGXSXEOCU
|
6.2 | Ki | 24 | — | |
XOVPCPRZRHQFBI
|
6.2 | Ki | 15 | — | |
YKYRQCWLYUTVIE
|
6.2 | Ki | 16 | — | |
ZGZVRPRSFXRGCF
|
6.2 | Ki | 76 | — | |
BDMXFIMYKGLQAL
|
6.2 | IC50 | 9 | — | |
DYIOAOFYWZXKEX
|
6.2 | IC50 | 4 | — | |
DYIOAOFYWZXKEX
|
6.2 | IC50 | 4 | — | |
MXIKVRCYCKFUND
|
6.2 | IC50 | 6 | — | |
FIVWKNZKXNNFCW
|
6.2 | IC50 | 9 | — | |
OGPJOAYIAOEJAM
|
6.2 | IC50 | 8 | — | |
BWORFRWIDWQHPL
|
6.2 | IC50 | 7 | — | |
DJHMDVUOYUYLOJ
|
6.2 | IC50 | 9 | — | |
KQZBWTMAFLOSPA
|
6.2 | IC50 | 8 | — | |
QVLJVHWQAKYGQI
|
6.2 | IC50 | 8 | — | |
IRBWROIEALHOPH
|
6.2 | IC50 | 7 | — | |
MQRHLOPPMRFMKM
|
6.2 | IC50 | 9 | — | |
PPQSZAVBAJMLRF
|
6.2 | IC50 | 5 | — | |
VGWCJGBQHCMHNJ
|
6.2 | IC50 | 8 | — | |
WHPORTUXBLFUPA
|
6.2 | IC50 | 8 | — | |
WVXNSAVVKYZVOE
|
6.2 | IC50 | 92 | — | |
RUQXGVGYNKIGJD
|
6.1 | IC50 | 7 | — | |
XXIXFZAUCITSCM
|
6.1 | IC50 | 7 | — | |
YRFAWSIUIFNVQA
|
6.1 | IC50 | 9 | — | |
HBBPDNLIBIZZFL
|
6.1 | IC50 | 7 | — | |
WHPORTUXBLFUPA
|
6.1 | IC50 | 9 | — | |
YDTHCIZMSQZYMR
|
6.1 | IC50 | 9 | — | |
BXNJHAXVSOCGBA
|
6.1 | IC50 | 14 | — | |
CPGKMMMSMJKHDL
|
6.1 | Ki | 16 | — |