Target Details
| UniProt AC | O43781 |
|---|---|
| Gene Symbol | DYRK3 |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 301
- Clinical molecules 4
- Avg pChEMBL 6.64
Active Molecules (301)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ROPFCXUWNMYMSW
|
6.5 | IC50 | 10 | — | |
RYWACTNAXCMTTN
|
6.5 | IC50 | 9 | — | |
YSBCFQVEEKUZSU
|
6.5 | IC50 | 9 | — | |
AOGIFFVMTGMFBP
|
6.5 | IC50 | 8 | — | |
JBWDTSLHUJHODF
|
6.4 | IC50 | 9 | — | |
JBWDTSLHUJHODF
|
6.4 | IC50 | 9 | — | |
PRJNNPMIUGYOST
|
6.4 | IC50 | 14 | — | |
QTRZNDLLYHSJSH
|
6.4 | IC50 | 9 | — | |
KCTCLVINURCCIL
|
6.4 | IC50 | 7 | — | |
CALAEFSQWBJMDU
|
6.4 | Ki | 21 | — | |
FLEAYYMORDPWAJ
|
6.4 | Ki | 90 | — | |
KAKGFGCTONHQJW
|
6.4 | Ki | 25 | — | |
PGPHHJBZEGSUNE
|
6.4 | IC50 | 4 | — | |
PQNWNVWJXPSZFR
|
6.4 | Ki | 21 | — | |
QNWARURWFRZNNO
|
6.4 | IC50 | 7 | — | |
RLTCEYSNDOXWKS
|
6.4 | IC50 | 9 | — | |
SGHXFHRRWFLILP
|
6.4 | Ki | 29 | — | |
YORVMWUGDVGXOQ
|
6.4 | IC50 | 8 | — | |
HFLXYSRIPKXGOQ
|
6.4 | IC50 | 4 | — | |
QVYXLOYBJBMXNP
|
6.4 | IC50 | 7 | — | |
VDJFUWZMISVQGO
|
6.4 | IC50 | 4 | — | |
DYHKEGKDOOZETF
|
6.4 | IC50 | 9 | — | |
JDNVNTCGESXSFD
|
6.4 | IC50 | 4 | — | |
QTRZNDLLYHSJSH
|
6.4 | IC50 | 9 | — | |
GVANUSPDJMCBIK
|
6.4 | IC50 | 6 | — | |
OYDWEMSWMQKSLK
|
6.4 | IC50 | 8 | — | |
HGMCNIGKEVZHFM
|
6.3 | IC50 | 8 | — | |
HMDPCTZKMDHQTP
|
6.3 | IC50 | 5 | — | |
AMBKAVGTUWUVBS
|
6.3 | IC50 | 8 | — | |
OHARPIGKJAKOCM
|
6.3 | IC50 | 8 | — | |
MIEPXFZAJZPNFG
|
6.3 | IC50 | 5 | — | |
MIEPXFZAJZPNFG
|
6.3 | IC50 | 8 | — | |
BWKADHBOXYDZFU
|
6.3 | IC50 | 10 | — | |
CBTNARFZVOPLBO
|
6.3 | IC50 | 5 | — | |
DOWFKLSBHHHHTF
|
6.3 | IC50 | 4 | — | |
QCHDHJOEPUQALZ
|
6.3 | IC50 | 9 | — | |
WREJZZXSNOJGIW
|
6.3 | IC50 | 9 | — | |
JWQOJVOKBAAAAR
|
6.3 | Ki | 29 | — | |
LRINYHMQZRENCY
|
6.3 | Ki | 29 | — | |
OQSBQXVIMQMCES
|
6.3 | IC50 | 9 | — | |
PNKALLUVKOKYHZ
|
6.3 | Ki | 32 | — | |
QONPPIZSNSSCSK
|
6.3 | Ki | 45 | Yes | |
RFVBRKXQYUDGIO
|
6.3 | Ki | 23 | — | |
RUQXGVGYNKIGJD
|
6.3 | IC50 | 9 | — | |
SVUIYNKSDCANAY
|
6.3 | Ki | 16 | — | |
XBNSDTLFWKORGH
|
6.3 | Ki | 10 | — | |
BBCSUMURJUYILA
|
6.3 | IC50 | 10 | — | |
JANQPHRPUAYQTA
|
6.3 | IC50 | 5 | — | |
WSUWIXYPBRLNOT
|
6.3 | IC50 | 4 | — | |
FBURYRMHEHTVED
|
6.3 | IC50 | 9 | — |