Target Details
| UniProt AC | O43781 |
|---|---|
| Gene Symbol | DYRK3 |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 301
- Clinical molecules 4
- Avg pChEMBL 6.64
Active Molecules (301)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LZUJDIWVWSRLRQ
|
6.7 | IC50 | 4 | — | |
LZUJDIWVWSRLRQ
|
6.7 | IC50 | 4 | — | |
UTFXYGYVDDLJER
|
6.7 | Ki | 36 | — | |
VLEFVPMCVJDTHZ
|
6.7 | Ki | 13 | — | |
XJJYJNMNYDNXNO
|
6.7 | Ki | 23 | — | |
XMFUGSRATNLPRM
|
6.7 | Ki | 19 | — | |
XYZNKCSDQRKAFR
|
6.7 | Ki | 53 | — | |
GXCOUFPTCZUTEE
|
6.7 | IC50 | 10 | — | |
DXVSNYWBRDTHFF
|
6.7 | IC50 | 10 | — | |
SBYPANVVFZBWDF
|
6.7 | IC50 | 9 | — | |
ZFOMCSNUEHMROO
|
6.7 | IC50 | 7 | — | |
FIVWKNZKXNNFCW
|
6.6 | IC50 | 8 | — | |
RGKOSKZCLZXDJI
|
6.6 | IC50 | 4 | — | |
WKYMGORXOQPTTO
|
6.6 | IC50 | 9 | — | |
BPNUQXPIQBZCMR
|
6.6 | Ki | 60 | — | |
KNVOICXEDILAGT
|
6.6 | Ki | 17 | — | |
LXVBELDBJGYFEM
|
6.6 | Ki | 20 | — | |
LYNBNVBMAGDJRW
|
6.6 | Ki | 81 | — | |
ORUUEFDGYYTXAF
|
6.6 | Ki | 26 | — | |
TWCARTFPHQNBPF
|
6.6 | Ki | 16 | — | |
PGPHHJBZEGSUNE
|
6.6 | IC50 | 21 | — | |
YHZQZEGQCKWCLP
|
6.6 | IC50 | 9 | — | |
HJEKFRDOAYXXRU
|
6.5 | IC50 | 8 | — | |
OVVHFDIQCYTOAS
|
6.5 | IC50 | 9 | — | |
NZMFVJNZGKELJC
|
6.5 | IC50 | 4 | — | |
SJYQOVMGZOATNK
|
6.5 | IC50 | 9 | — | |
USYASDQVUTWEQM
|
6.5 | IC50 | 9 | — | |
YAXGFAAKCUOWNM
|
6.5 | IC50 | 9 | — | |
CHQYAWLKOUOTQO
|
6.5 | IC50 | 20 | — | |
FANUXQYVRUHAAH
|
6.5 | IC50 | 6 | — | |
QCTMVDQWYGRUJK
|
6.5 | IC50 | 9 | — | |
FJAIARRQBXWUMX
|
6.5 | IC50 | 2 | — | |
GDYZFFBMSBDTAA
|
6.5 | Ki | 60 | — | |
ITOTZLBIDAOTGK
|
6.5 | IC50 | 4 | — | |
IUEBPIPDFMCSTP
|
6.5 | Ki | 29 | — | |
KRIUNPBAQZGFQA
|
6.5 | Ki | 76 | — | |
UEIRKXUBXCSHJE
|
6.5 | Ki | 19 | — | |
VBYRFFCBZNEHAL
|
6.5 | IC50 | 4 | — | |
YMIJUBCSOKSFRU
|
6.5 | Ki | 87 | — | |
ZGDSBEUMPIMXBM
|
6.5 | Ki | 42 | — | |
BBCSUMURJUYILA
|
6.5 | IC50 | 9 | — | |
ITOTZLBIDAOTGK
|
6.5 | IC50 | 4 | — | |
PGPHHJBZEGSUNE
|
6.5 | IC50 | 17 | — | |
ZBKFRVXDYILXFJ
|
6.5 | IC50 | 6 | — | |
WFOMWAYINPJPDX
|
6.5 | IC50 | 9 | — | |
LVSVYVPFNYRNOF
|
6.5 | IC50 | 8 | — | |
YSODDCRKIDDXKM
|
6.5 | IC50 | 9 | — | |
BEILWJKGWBDPRG
|
6.5 | IC50 | 7 | — | |
GEJSQZULGDKBQV
|
6.5 | IC50 | 8 | — | |
KRXQWLCJHMDEDM
|
6.5 | IC50 | 8 | — |