Target Details
| UniProt AC | O43781 |
|---|---|
| Gene Symbol | DYRK3 |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 301
- Clinical molecules 4
- Avg pChEMBL 6.64
Active Molecules (301)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SLKHMZQUNIHINK
|
7.2 | IC50 | 10 | — | |
GDSQVLMYYCNAGP
|
7.2 | IC50 | 6 | — | |
YJKPCYDSZXIODK
|
7.1 | IC50 | 8 | — | |
FPQHXFMYXQZPSV
|
7.1 | Ki | 23 | — | |
GHAZVJQMLWOQLP
|
7.1 | Ki | 17 | — | |
MVJMMLFMPWITEJ
|
7.1 | Ki | 110 | — | |
NRSGWEVTVGZDFC
|
7.1 | Ki | 50 | — | |
OWFLADWRSCINST
|
7.1 | Ki | 30 | — | |
KAGWQDFFFLWBFD
|
7.1 | IC50 | 8 | — | |
GCSZJMUFYOAHFY
|
7.1 | IC50 | 8 | — | |
QSGKPYRFWJINEH
|
7.0 | IC50 | 12 | — | |
CWJLAVRXVFHDSJ
|
7.0 | IC50 | 13 | — | |
DFMCXVONDDGQIY
|
7.0 | Ki | 66 | — | |
KAICHBSRWFIESE
|
7.0 | Ki | 14 | — | |
LRZYYIZFBXFSJB
|
7.0 | Ki | 69 | — | |
MASJMHFQMYAPJR
|
7.0 | Ki | 41 | — | |
DSCUTYQYWCTFQL
|
7.0 | IC50 | 6 | — | |
YGXHQYJKJUFSJI
|
7.0 | IC50 | 14 | — | |
OWDVXJJCVWTPPW
|
7.0 | IC50 | 8 | — | |
PBGPFWACZLCJFH
|
7.0 | IC50 | 3 | — | |
SJWUVVGOTOMGOH
|
6.9 | IC50 | 9 | — | |
CQZSVQKINMHLBO
|
6.9 | IC50 | 4 | — | |
DCJOTKUJWJFCSP
|
6.9 | IC50 | 9 | — | |
UUXDJIVNVOOKFQ
|
6.9 | IC50 | 9 | — | |
JFDRONLMXPRQPP
|
6.9 | IC50 | 9 | — | |
GHMRUNOHAHJNNA
|
6.9 | Ki | 29 | — | |
KYACBMRLQMEIAI
|
6.9 | Ki | 30 | — | |
OWDRQHVEJIYVOI
|
6.9 | Ki | 47 | — | |
SBFPHSVZEXSHTL
|
6.9 | Ki | 62 | — | |
SYLTYCLPHHSEIJ
|
6.9 | Ki | 27 | — | |
XCHWBXBDZRJVDP
|
6.9 | Ki | 51 | — | |
XPHWIERLJBFPFV
|
6.9 | Ki | 69 | — | |
SKKBUBMBPCJYKW
|
6.9 | IC50 | 9 | — | |
IJFKKIMDRSZOOW
|
6.9 | IC50 | 9 | — | |
KYOPCGIPHGGWMV
|
6.8 | IC50 | 7 | — | |
UTDNMHFLZJFPPY
|
6.8 | IC50 | 4 | — | |
VRGNMDTYOWQXQC
|
6.8 | IC50 | 8 | — | |
VRGNMDTYOWQXQC
|
6.8 | IC50 | 5 | — | |
GCBJDOWIQHMCMR
|
6.8 | Ki | 84 | — | |
MIKAKZKNMYZLDX
|
6.8 | Ki | 42 | — | |
OHPRWVPOPFGLJG
|
6.8 | Ki | 19 | — | |
QEWSTOOMTBAUAG
|
6.8 | Ki | 17 | — | |
QXMXIHBLICGPMG
|
6.8 | IC50 | 9 | — | |
SQXSMLLCDWJNAC
|
6.8 | Ki | 20 | — | |
UBUJLBVNZCRWPX
|
6.8 | IC50 | 7 | — | |
AKNIGLLNHUTMPO
|
6.8 | IC50 | 9 | — | |
ZBYBDKHFLSHGBP
|
6.8 | IC50 | 4 | — | |
ZBYBDKHFLSHGBP
|
6.7 | IC50 | 4 | — | |
CBTNARFZVOPLBO
|
6.7 | IC50 | 8 | — | |
CZIGMBNEFWBEMD
|
6.7 | Ki | 16 | — |