Target Details
| UniProt AC | O43781 |
|---|---|
| Gene Symbol | DYRK3 |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 301
- Clinical molecules 4
- Avg pChEMBL 6.64
Active Molecules (301)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IUWWRSQCDUQDEZ
|
10.0 | IC50 | 8 | — | |
IUWWRSQCDUQDEZ
|
10.0 | IC50 | 9 | — | |
VCTLOEWZYIGVBO
|
8.7 | IC50 | 12 | — | |
FUMCKNCUEAQHCV
|
8.3 | Ki | 103 | — | |
NJPWCTYVEJIQBM
|
8.3 | Ki | 72 | — | |
BSFNGHCTZDCQBF
|
8.1 | Ki | 93 | — | |
CLEGDJQQHUTCOW
|
8.1 | Ki | 43 | — | |
RJZDECGDCKOHBV
|
8.1 | Ki | 70 | — | |
CHTMRWQLNNRRFJ
|
8.0 | Ki | 70 | — | |
JJJSCYSPSKBQAX
|
8.0 | Ki | 34 | — | |
RKUKAACYUCUJEE
|
8.0 | Ki | 58 | — | |
YEZMGVBTPDYRPO
|
8.0 | IC50 | 8 | — | |
QTHCAAFKVUWAFI
|
8.0 | IC50 | 23 | — | |
QIYXLIZWXGGKOO
|
7.9 | IC50 | 10 | — | |
DPDVVGCNUWGGRS
|
7.8 | IC50 | 10 | — | |
NBTJWRPKGNQBJS
|
7.8 | IC50 | 8 | — | |
QAJPIJHWTGPUNZ
|
7.8 | Ki | 37 | — | |
MNVPCONHWCXDES
|
7.8 | IC50 | 9 | — | |
HKSZLNNOFSGOKW
|
7.8 | IC50 | 408 | — | |
HEVBCYZPXGZFGS
|
7.7 | IC50 | 11 | — | |
UZWDCWONPYILKI
|
7.7 | IC50 | 47 | — | |
RYBNARZBIXTFJS
|
7.7 | IC50 | 9 | — | |
RYBNARZBIXTFJS
|
7.7 | IC50 | 9 | — | |
QMUKOEKTUBVPFU
|
7.7 | IC50 | 12 | — | |
CGRDYMCBGXJNLR
|
7.6 | IC50 | 9 | — | |
BWNQBFHVFFZHMR
|
7.6 | IC50 | 10 | — | |
QXFBTYPBHYOEMX
|
7.6 | IC50 | 9 | — | |
RJYLSCSDDDQEPD
|
7.6 | IC50 | 10 | — | |
ZYTFPHRVOZXPGZ
|
7.6 | Ki | 30 | — | |
SJWUVVGOTOMGOH
|
7.5 | IC50 | 10 | — | |
MGEGGAFJSKMJJD
|
7.5 | IC50 | 5 | — | |
VCFPJHJKTXRDGD
|
7.5 | IC50 | 3 | — | |
MUOKSQABCJCOPU
|
7.5 | IC50 | 36 | — | |
VMOVZKURWYNTLN
|
7.5 | Ki | 7 | — | |
VXYDJXMHISGSDA
|
7.5 | Ki | 59 | — | |
CGPYAXSYKQBYKJ
|
7.5 | IC50 | 12 | — | |
BUDHVVXPBGMAPV
|
7.4 | IC50 | 11 | — | |
SJWUVVGOTOMGOH
|
7.4 | IC50 | 12 | — | |
CIICGXXZCWRFQE
|
7.4 | IC50 | 7 | — | |
CLRFYTGANQZOBS
|
7.4 | Ki | 41 | — | |
KHVQTEBOVFILCQ
|
7.4 | IC50 | 10 | — | |
FGBSSPMQGRUJPS
|
7.3 | IC50 | 10 | — | |
KBMQGIPVJGXLOU
|
7.3 | IC50 | 7 | — | |
DKXHSOUZPMHNIZ
|
7.3 | Ki | 51 | Yes | |
DYSRECIVMDGUQU
|
7.3 | Ki | 29 | — | |
OUJZYQBEFNDJQN
|
7.3 | Ki | 71 | — | |
RJXWGPDMMDILGJ
|
7.3 | IC50 | 9 | — | |
UGYUFJPHSWYELP
|
7.2 | IC50 | 8 | — | |
ADMFLILDQJSEIK
|
7.2 | Ki | 72 | — | |
XFWUTMHVDGPWLH
|
7.2 | Ki | 75 | — |