Target Details
| UniProt AC | O43683 |
|---|---|
| Gene Symbol | BUB1 |
| Protein Name | Mitotic checkpoint serine/threonine-protein kinase BUB1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08311 (Mad3_BUB1_I) PF00069 (Pkinase) |
Summary
- Multi-target molecules 14
- Clinical molecules 3
- Avg pChEMBL 7.05
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (14)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QVOGVAVHOLLLAZ
|
8.5 | IC50 | 4 | — | |
CAOVBAQHBWKZJG
|
7.8 | IC50 | 3 | — | |
OEXTZXWPZXNIIH
|
7.7 | IC50 | 3 | — | |
BSAVGANXIAKUQK
|
7.7 | IC50 | 3 | — | |
BSAVGANXIAKUQK
|
7.7 | IC50 | 3 | — | |
LPYBJNPKBPALQQ
|
7.6 | IC50 | 3 | — | |
MWKSRKSEWLRPBL
|
7.1 | Kd | 1075 | — | |
LOLPPWBBNUVNQZ
|
7.0 | Kd | 97 | Yes | |
AAKJLRGGTJKAMG
|
7.0 | Kd | 50 | Yes | |
FPQNRXITKTZFMF
|
6.6 | Kd | 13 | — | |
PLIVFNIUGLLCEK
|
6.0 | Kd | 20 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |