Target Details
| UniProt AC | O43614 |
|---|---|
| Gene Symbol | HCRTR2 |
| Protein Name | Orexin receptor type 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) PF03827 (Orexin_rec2) |
Summary
- Multi-target molecules 3,873
- Clinical molecules 0
- Avg pChEMBL 7.34
KEGG Pathways (2)
Active Molecules (3,873)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RHUPJZFHSQTXAK
|
9.0 | IC50 | 2 | — | |
RRGQDAPENZQDHE
|
9.0 | IC50 | 2 | — | |
RZIWRUCHHJWXCX
|
9.0 | IC50 | 2 | — | |
SGCLCURYCKUVAD
|
9.0 | IC50 | 2 | — | |
TVOPOIUNCIFOAI
|
9.0 | IC50 | 2 | — | |
UCGAGGJWCWXTIP
|
9.0 | IC50 | 2 | — | |
URIHGJROOMIUNL
|
9.0 | IC50 | 2 | — | |
VDPZWYVAUUMDAS
|
9.0 | Ki | 2 | — | |
VPGMOJNQLSGSJB
|
9.0 | IC50 | 2 | — | |
WLBCPTKNCBIYOL
|
9.0 | IC50 | 2 | — | |
WMNXZVYJHQFMCI
|
9.0 | Ki | 2 | — | |
WMSOKWMKDYBMFL
|
9.0 | IC50 | 2 | — | |
WRPGNWQVJUWOTB
|
9.0 | Ki | 2 | — | |
WYKNCJASXYZRBP
|
9.0 | IC50 | 2 | — | |
XBKLSMQHNWPYAS
|
9.0 | IC50 | 2 | — | |
XVMBACKIQPNUGC
|
9.0 | IC50 | 2 | — | |
ZGXURSBUSGZSFT
|
9.0 | IC50 | 2 | — | |
KJPHTXTWFHVJIG
|
9.0 | Ki | 2 | — | |
KJPHTXTWFHVJIG
|
9.0 | Ki | 2 | — | |
KJPHTXTWFHVJIG
|
9.0 | Ki | 2 | — | |
PHPUKRNBBIXYQK
|
9.0 | IC50 | 2 | — | |
ARTAPIITUFBDOM
|
8.9 | Ki | 2 | — | |
GVNLLQCJDVUODJ
|
8.9 | IC50 | 2 | — | |
WCUGLZXLNMVHNW
|
8.9 | Ki | 2 | — | |
AEZZJXJIJFSUEM
|
8.9 | IC50 | 2 | — | |
IQBQPKYTEMWHQG
|
8.9 | IC50 | 2 | — | |
NUSPCNSRGWNZOD
|
8.9 | IC50 | 2 | — | |
XBPCRHBKTGGYRS
|
8.9 | IC50 | 2 | — | |
XMTCRKRHFLBROW
|
8.9 | IC50 | 2 | — | |
AEZZJXJIJFSUEM
|
8.9 | IC50 | 2 | — | |
VTGVYRYFFCPVDP
|
8.9 | Ki | 2 | — | |
BVUZOFDSUCGTDO
|
8.9 | Ki | 2 | — | |
HCBUJXNAUZXQJZ
|
8.9 | Ki | 2 | — | |
LIHWSYUGQWXXBX
|
8.9 | IC50 | 2 | — | |
WEPOQCBGFBAHKW
|
8.9 | IC50 | 2 | — | |
ZLGOHPFJEPYOQA
|
8.9 | IC50 | 2 | — | |
HIYMXVSQZFCQBY
|
8.8 | Ki | 2 | — | |
JOCIBZPBSCTMTE
|
8.8 | IC50 | 2 | — | |
OIYSQHUALQGVNP
|
8.8 | IC50 | 2 | — | |
WDQKCMWGNYOTEG
|
8.8 | IC50 | 2 | — | |
BTYVZVITBHYSBW
|
8.8 | IC50 | 2 | — | |
NNYOYMBIEDPXHF
|
8.8 | IC50 | 2 | — | |
DGCYMZXGGJWTPE
|
8.8 | IC50 | 2 | — | |
DUNPFBVKEJBJDW
|
8.8 | IC50 | 2 | — | |
FOEWIXNBXKVERV
|
8.8 | Ki | 2 | — | |
GGEFNKYUDAADPY
|
8.8 | IC50 | 2 | — | |
NADVAWWMPXTUET
|
8.8 | Ki | 2 | — | |
QRWIMPDPKYXNEE
|
8.8 | Ki | 2 | — | |
UCTMYARPCLQYDJ
|
8.8 | IC50 | 2 | — | |
ZVQWWVVTWJLQAK
|
8.8 | Ki | 2 | — |