Target Details
| UniProt AC | O43613 |
|---|---|
| Gene Symbol | HCRTR1 |
| Protein Name | Orexin/Hypocretin receptor type 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 3,881
- Clinical molecules 0
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (3,881)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NFCVBPAPRRTXCA
|
8.4 | Ki | 2 | — | |
NFCVBPAPRRTXCA
|
8.4 | Ki | 2 | — | |
NTNSUMPZQLAAMK
|
8.4 | IC50 | 2 | — | |
ODRSUBOCIUQDQX
|
8.4 | IC50 | 2 | — | |
OESAAULEOZNLQH
|
8.4 | IC50 | 2 | — | |
OFOKYTZDYMGETB
|
8.4 | IC50 | 2 | — | |
OIOSLKQRWPKHHK
|
8.4 | IC50 | 2 | — | |
OJVPFTHFYQCMAZ
|
8.4 | IC50 | 2 | — | |
OLGPONWRXCYWQO
|
8.4 | IC50 | 2 | — | |
ORPRTCJZBDNPEM
|
8.4 | IC50 | 2 | — | |
ORWFLSUKJBCAEL
|
8.4 | IC50 | 2 | — | |
OWFVNBHKYXWMAX
|
8.4 | Kd | 2 | — | |
PCPHRHBXQANSIF
|
8.4 | IC50 | 2 | — | |
PGRFCBWNHDMEMV
|
8.4 | Ki | 2 | — | |
PMLWCCOLXOVHLE
|
8.4 | IC50 | 2 | — | |
PXDWETVKDHRZFI
|
8.4 | Ki | 2 | — | |
QHOOFEYVMVIMAH
|
8.4 | IC50 | 2 | — | |
QOZHEUNRUWRYRC
|
8.4 | Ki | 2 | — | |
QQRIUHPUFYGSTQ
|
8.4 | IC50 | 2 | — | |
QWHXRHHISYFFAY
|
8.4 | Ki | 2 | — | |
RKLPQCPZHKBFPB
|
8.4 | IC50 | 2 | — | |
RSCBRJAESFFMDG
|
8.4 | IC50 | 2 | — | |
RSXSJNWYISSNHS
|
8.4 | IC50 | 2 | — | |
RVFWGCRTBRYICQ
|
8.4 | IC50 | 2 | — | |
SEIYMHWXOQHIRD
|
8.4 | IC50 | 2 | — | |
SMVHMTBUOLIQMT
|
8.4 | IC50 | 2 | — | |
STCNMOVPLMYXAN
|
8.4 | IC50 | 2 | — | |
TXOLBWQUYQXATH
|
8.4 | IC50 | 2 | — | |
UCGAGGJWCWXTIP
|
8.4 | IC50 | 2 | — | |
UCYBAXWWBPSWIL
|
8.4 | IC50 | 2 | — | |
UXOGHIYIIAOJFE
|
8.4 | IC50 | 2 | — | |
VXKUPARUVUBAQK
|
8.4 | IC50 | 2 | — | |
WLGKPVICVODJNZ
|
8.4 | IC50 | 2 | — | |
WYPLVRJYHWKAPV
|
8.4 | Ki | 2 | — | |
XICYINDZEAEGIE
|
8.4 | IC50 | 2 | — | |
YEGSYMNMIHXAMS
|
8.4 | IC50 | 2 | — | |
YRDYMMSFSGXWLF
|
8.4 | IC50 | 2 | — | |
ZACJKMOEFBPFHF
|
8.4 | Ki | 2 | — | |
ZRQPVUWXLKQQII
|
8.4 | IC50 | 2 | — | |
AGUKCTFKQWNLSC
|
8.4 | IC50 | 2 | — | |
JAZZMBNYLJZYMJ
|
8.4 | Ki | 2 | — | |
NHRZLARRAZSSNB
|
8.4 | IC50 | 2 | — | |
AFXBOTJWXUOBKK
|
8.4 | IC50 | 2 | — | |
CHLAMJXRDIVYQK
|
8.4 | Ki | 2 | — | |
JNJOBZPIHMXOSP
|
8.4 | IC50 | 2 | — | |
MLMWHEAQEAOHLI
|
8.4 | IC50 | 2 | — | |
NUSPCNSRGWNZOD
|
8.4 | IC50 | 2 | — | |
VFSSJHGGWPJHRS
|
8.4 | IC50 | 2 | — | |
DLINKHARPOJPKX
|
8.3 | IC50 | 2 | — | |
GTAYPYFUGIRKPJ
|
8.3 | IC50 | 2 | — |