Target Details
| UniProt AC | O43613 |
|---|---|
| Gene Symbol | HCRTR1 |
| Protein Name | Orexin/Hypocretin receptor type 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 3,881
- Clinical molecules 0
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (3,881)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OKROKECXNXWALA
|
8.5 | IC50 | 2 | — | |
GUQHPENKNGCHKL
|
8.4 | IC50 | 2 | — | |
HZJTWMIUOYBHLN
|
8.4 | IC50 | 2 | — | |
JPORFXWIBQIBLN
|
8.4 | IC50 | 2 | — | |
MASVQPOUODOSNG
|
8.4 | IC50 | 2 | — | |
OGRBDFWIZPXZCZ
|
8.4 | IC50 | 2 | — | |
OMTPFVJZEZVSIP
|
8.4 | IC50 | 2 | — | |
XOEICXYQCMGMQQ
|
8.4 | IC50 | 2 | — | |
VWFHAQXJYLRSEX
|
8.4 | IC50 | 2 | — | |
HCUREBSNYDMSKO
|
8.4 | IC50 | 2 | — | |
IBJBAQDMTLBIEQ
|
8.4 | IC50 | 2 | — | |
PUZZWRPQBVSLOP
|
8.4 | IC50 | 2 | — | |
HYBZWVLPALMACV
|
8.4 | Ki | 4 | — | |
KNSSBXCHRPNPDS
|
8.4 | Kd | 2 | — | |
AFSCYCXJAKZMAT
|
8.4 | IC50 | 2 | — | |
APOGCVQZYGMWMJ
|
8.4 | IC50 | 2 | — | |
ARSBQKPKEHFSQL
|
8.4 | Ki | 2 | — | |
BXNCXMMOWAUHNN
|
8.4 | IC50 | 2 | — | |
CDBNZCXRTRXXQF
|
8.4 | IC50 | 2 | — | |
CEFZLJAZLPOVTE
|
8.4 | Ki | 2 | — | |
CILYBMUJEDXLPI
|
8.4 | IC50 | 2 | — | |
CLOOLVHJLDFMDV
|
8.4 | IC50 | 2 | — | |
CNCDUEDPGAHZTP
|
8.4 | IC50 | 2 | — | |
CXUTWSQJWLDTGV
|
8.4 | IC50 | 2 | — | |
DBDQRJSDHDMDBC
|
8.4 | IC50 | 2 | — | |
FCYJFENZGHEDRB
|
8.4 | IC50 | 2 | — | |
FXEJYJOLEHLEJH
|
8.4 | IC50 | 2 | — | |
GFECZBYZFVWZHJ
|
8.4 | Ki | 2 | — | |
GJIDHTCQPKWTIL
|
8.4 | IC50 | 2 | — | |
HKYJQQKWZCIZNH
|
8.4 | Ki | 2 | — | |
HYFRBSMLWUEXKY
|
8.4 | IC50 | 2 | — | |
HYSRABRBUHZYQJ
|
8.4 | IC50 | 2 | — | |
IIVBMGSJEAWDEA
|
8.4 | Ki | 2 | — | |
IKRKJQANDJSOOF
|
8.4 | Ki | 2 | — | |
IUICMZGKDMRYTR
|
8.4 | Kd | 2 | — | |
JNZNQAZDCIXPAH
|
8.4 | IC50 | 2 | — | |
JSJSRBOREVOTHH
|
8.4 | IC50 | 2 | — | |
JVZPIDIYRSKRCP
|
8.4 | IC50 | 2 | — | |
KBOYUJJQCAMZDT
|
8.4 | Ki | 2 | — | |
KYJDZVZDSWHGJA
|
8.4 | IC50 | 2 | — | |
LEGFFCFGSFQDHY
|
8.4 | IC50 | 2 | — | |
LFVHMZKMNVGVDF
|
8.4 | IC50 | 2 | — | |
LFWWMTWFACWYES
|
8.4 | Ki | 2 | — | |
LLMHHQJUBHBUPE
|
8.4 | IC50 | 2 | — | |
LZIZZUSWJHWVCS
|
8.4 | IC50 | 2 | — | |
LZTASGJPADXFHY
|
8.4 | IC50 | 2 | — | |
MEVYEKMBSZIAIZ
|
8.4 | IC50 | 2 | — | |
MFXXQQRKFPRHSL
|
8.4 | Ki | 2 | — | |
MYSKBZWJKAYHAI
|
8.4 | IC50 | 2 | — | |
MYYWNWGKGXQLPB
|
8.4 | IC50 | 2 | — |