Target Details
UniProt ACO43613
Gene SymbolHCRTR1
Protein NameOrexin/Hypocretin receptor type 1
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 3,881
  • Clinical molecules 0
  • Avg pChEMBL 7.32
Top Co-occurrence Targets
Active Molecules (3,881)
InChIKey pChEMBL Type Targets Clinical
OKROKECXNXWALA 8.5 IC50 2
GUQHPENKNGCHKL 8.4 IC50 2
HZJTWMIUOYBHLN 8.4 IC50 2
JPORFXWIBQIBLN 8.4 IC50 2
MASVQPOUODOSNG 8.4 IC50 2
OGRBDFWIZPXZCZ 8.4 IC50 2
OMTPFVJZEZVSIP 8.4 IC50 2
XOEICXYQCMGMQQ 8.4 IC50 2
VWFHAQXJYLRSEX 8.4 IC50 2
HCUREBSNYDMSKO 8.4 IC50 2
IBJBAQDMTLBIEQ 8.4 IC50 2
PUZZWRPQBVSLOP 8.4 IC50 2
HYBZWVLPALMACV 8.4 Ki 4
KNSSBXCHRPNPDS 8.4 Kd 2
AFSCYCXJAKZMAT 8.4 IC50 2
APOGCVQZYGMWMJ 8.4 IC50 2
ARSBQKPKEHFSQL 8.4 Ki 2
BXNCXMMOWAUHNN 8.4 IC50 2
CDBNZCXRTRXXQF 8.4 IC50 2
CEFZLJAZLPOVTE 8.4 Ki 2
CILYBMUJEDXLPI 8.4 IC50 2
CLOOLVHJLDFMDV 8.4 IC50 2
CNCDUEDPGAHZTP 8.4 IC50 2
CXUTWSQJWLDTGV 8.4 IC50 2
DBDQRJSDHDMDBC 8.4 IC50 2
FCYJFENZGHEDRB 8.4 IC50 2
FXEJYJOLEHLEJH 8.4 IC50 2
GFECZBYZFVWZHJ 8.4 Ki 2
GJIDHTCQPKWTIL 8.4 IC50 2
HKYJQQKWZCIZNH 8.4 Ki 2
HYFRBSMLWUEXKY 8.4 IC50 2
HYSRABRBUHZYQJ 8.4 IC50 2
IIVBMGSJEAWDEA 8.4 Ki 2
IKRKJQANDJSOOF 8.4 Ki 2
IUICMZGKDMRYTR 8.4 Kd 2
JNZNQAZDCIXPAH 8.4 IC50 2
JSJSRBOREVOTHH 8.4 IC50 2
JVZPIDIYRSKRCP 8.4 IC50 2
KBOYUJJQCAMZDT 8.4 Ki 2
KYJDZVZDSWHGJA 8.4 IC50 2
LEGFFCFGSFQDHY 8.4 IC50 2
LFVHMZKMNVGVDF 8.4 IC50 2
LFWWMTWFACWYES 8.4 Ki 2
LLMHHQJUBHBUPE 8.4 IC50 2
LZIZZUSWJHWVCS 8.4 IC50 2
LZTASGJPADXFHY 8.4 IC50 2
MEVYEKMBSZIAIZ 8.4 IC50 2
MFXXQQRKFPRHSL 8.4 Ki 2
MYSKBZWJKAYHAI 8.4 IC50 2
MYYWNWGKGXQLPB 8.4 IC50 2
2D structure