Target Details
| UniProt AC | O43613 |
|---|---|
| Gene Symbol | HCRTR1 |
| Protein Name | Orexin/Hypocretin receptor type 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 3,881
- Clinical molecules 0
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (3,881)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QIKVTMHZHYXNDE
|
8.5 | IC50 | 2 | — | |
QNFGBHOABLCVGZ
|
8.5 | IC50 | 2 | — | |
RKLPQCPZHKBFPB
|
8.5 | IC50 | 2 | — | |
SDUCADJXPVQZIE
|
8.5 | Ki | 2 | — | |
SKRGGMWIJIAQDK
|
8.5 | IC50 | 2 | — | |
TWMWEJVSFZPUFN
|
8.5 | Ki | 2 | — | |
UHZXDUKWSARABK
|
8.5 | IC50 | 2 | — | |
UIELPQGRXTWUBL
|
8.5 | IC50 | 2 | — | |
UXINVWZBFDJHKA
|
8.5 | IC50 | 2 | — | |
VKJYSIARVKDYIT
|
8.5 | IC50 | 2 | — | |
VLUXTCAIDBDMPI
|
8.5 | IC50 | 2 | — | |
VMCVDMDKIAUUAU
|
8.5 | Ki | 2 | — | |
VNEMVCXDERLURH
|
8.5 | IC50 | 2 | — | |
VPQUBVYYWSMYEA
|
8.5 | IC50 | 2 | — | |
WAKGEROYRUJRJS
|
8.5 | IC50 | 2 | — | |
WDQKCMWGNYOTEG
|
8.5 | IC50 | 2 | — | |
WOMLJIMOFFDWMO
|
8.5 | IC50 | 2 | — | |
WRLVGTRMEZGZFE
|
8.5 | IC50 | 2 | — | |
WVPBMKQMORLKAZ
|
8.5 | IC50 | 2 | — | |
WVZLCGIQGDVCKB
|
8.5 | Ki | 2 | — | |
WYFQHYNFGVNXFG
|
8.5 | IC50 | 2 | — | |
XKKKABNXFDRANJ
|
8.5 | IC50 | 2 | — | |
XKUGHTYMIFCAQZ
|
8.5 | IC50 | 2 | — | |
XTIOBAAREREBIF
|
8.5 | IC50 | 2 | — | |
XYJCAEKTDPOHKG
|
8.5 | IC50 | 2 | — | |
YCPPLHONVRZFSC
|
8.5 | Ki | 2 | — | |
YCYUDFTUFUSQNS
|
8.5 | IC50 | 2 | — | |
YEDDEIUNRODXSF
|
8.5 | IC50 | 2 | — | |
YGNNSLBDINPURJ
|
8.5 | IC50 | 2 | — | |
YMXUVOVOEYJPGQ
|
8.5 | IC50 | 2 | — | |
YSBGRVXJEMSEQY
|
8.5 | Ki | 2 | — | |
MHBLBSQHRANVNC
|
8.5 | IC50 | 2 | — | |
DIUVTHBJFXAJNU
|
8.5 | Ki | 2 | — | |
FNSBFXNNFNCHOW
|
8.5 | Ki | 2 | — | |
PRTOIZDFTLVTTN
|
8.5 | Ki | 2 | — | |
FMDLORLPXIAIMQ
|
8.5 | IC50 | 2 | — | |
XMTCRKRHFLBROW
|
8.5 | IC50 | 2 | — | |
YZRHBGIKWQSFJJ
|
8.5 | IC50 | 2 | — | |
ZTYVXYZQICUWOW
|
8.5 | IC50 | 2 | — | |
ZYKKWUHUHNTMCV
|
8.5 | IC50 | 2 | — | |
JCHZZFRXFBKQHC
|
8.5 | IC50 | 2 | — | |
OMTCPGOATBMMKY
|
8.5 | IC50 | 2 | — | |
REIHLDGDOFIXTP
|
8.5 | IC50 | 2 | — | |
GJIDHTCQPKWTIL
|
8.5 | IC50 | 2 | — | |
LFPIOOYGMXHBRI
|
8.5 | IC50 | 2 | — | |
PXYCRNATPGCYAG
|
8.5 | IC50 | 2 | — | |
ATCMNCWZQLATOI
|
8.5 | IC50 | 2 | — | |
MPIPRURYZBEAQW
|
8.5 | Ki | 2 | — | |
MYRVFLCZPBNRHL
|
8.5 | IC50 | 2 | — | |
OIYSQHUALQGVNP
|
8.5 | IC50 | 2 | — |