Target Details
| UniProt AC | O43613 |
|---|---|
| Gene Symbol | HCRTR1 |
| Protein Name | Orexin/Hypocretin receptor type 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 3,881
- Clinical molecules 0
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (3,881)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SBDNJLCIYJRHKZ
|
8.7 | IC50 | 2 | — | |
SMWYFICPEVRFOB
|
8.7 | IC50 | 2 | — | |
STINWRWRNQHPGO
|
8.7 | IC50 | 2 | — | |
TWCRHJLMMAYSTE
|
8.7 | Ki | 3 | — | |
TYHOOCFBPYQMCS
|
8.7 | IC50 | 2 | — | |
TZVRPQFYZBQRPK
|
8.7 | IC50 | 2 | — | |
UNNYKAHMVYXHRC
|
8.7 | IC50 | 2 | — | |
UNRBBSQFBPJIAV
|
8.7 | IC50 | 2 | — | |
UNTSUUSNBKJZFC
|
8.7 | IC50 | 2 | — | |
VGFZJFYRKGSKGE
|
8.7 | IC50 | 2 | — | |
VGFZJFYRKGSKGE
|
8.7 | IC50 | 2 | — | |
WKXGFOWQJLVKST
|
8.7 | IC50 | 2 | — | |
WNICTQLZNYNDDE
|
8.7 | IC50 | 2 | — | |
XDAZJJGYLDZHNW
|
8.7 | IC50 | 2 | — | |
XDMPGWJRNRIXEC
|
8.7 | IC50 | 2 | — | |
XEYYOUAXMDVMSH
|
8.7 | Ki | 2 | — | |
XWVOVQAMOXFSHM
|
8.7 | IC50 | 2 | — | |
YNQCYKPXLIMHBV
|
8.7 | IC50 | 2 | — | |
YRVNCTCKYNIFSU
|
8.7 | IC50 | 2 | — | |
ZDGPOSKGUZNOIJ
|
8.7 | IC50 | 2 | — | |
ZESPBMRBBZNENN
|
8.7 | IC50 | 2 | — | |
ZTNQZEPNQJBTRM
|
8.7 | IC50 | 2 | — | |
ZXEWKIMFKPFZMU
|
8.7 | IC50 | 2 | — | |
ABQUTJKCXJRSSO
|
8.7 | IC50 | 2 | — | |
MAZDSKJURDSEEG
|
8.7 | Ki | 2 | — | |
AQFPGDOPAWNDQW
|
8.7 | IC50 | 2 | — | |
HIYMXVSQZFCQBY
|
8.7 | Ki | 2 | — | |
YZRHBGIKWQSFJJ
|
8.7 | IC50 | 2 | — | |
GGEFNKYUDAADPY
|
8.6 | IC50 | 2 | — | |
BZZDKUXANMBARX
|
8.6 | IC50 | 2 | — | |
FCVLRNRCGDIIDA
|
8.6 | IC50 | 2 | — | |
SRKVUFVTSRBFFN
|
8.6 | IC50 | 2 | — | |
SRKVUFVTSRBFFN
|
8.6 | IC50 | 2 | — | |
AIZXGTQGJBGNNH
|
8.6 | Ki | 2 | — | |
DGCYMZXGGJWTPE
|
8.6 | IC50 | 2 | — | |
LBOOMLHSTGFZSQ
|
8.6 | IC50 | 2 | — | |
NPFDWHQSDBWQLH
|
8.6 | Ki | 2 | — | |
XQNBEBURKKIKTM
|
8.6 | IC50 | 2 | — | |
XSAGNRRAVSAHPQ
|
8.6 | Ki | 2 | — | |
ZPLJPYAYQJTDJK
|
8.6 | Ki | 2 | — | |
LHSPBVKFWDHYSG
|
8.6 | IC50 | 2 | — | |
MPEBTPDHFLWMMX
|
8.6 | IC50 | 2 | — | |
SEIYMHWXOQHIRD
|
8.6 | IC50 | 2 | — | |
CWBJXWWFPDALKJ
|
8.6 | IC50 | 2 | — | |
FWHHRBMLQOYRQF
|
8.6 | IC50 | 2 | — | |
WQGLWMDRMSSGNV
|
8.6 | IC50 | 2 | — | |
PEAXRVOYMYUBCP
|
8.6 | IC50 | 2 | — | |
IFIYHYUCRGZDCI
|
8.5 | IC50 | 2 | — | |
JCFJSYCJOIPVJT
|
8.5 | IC50 | 2 | — | |
LSRYXWRLTUFERQ
|
8.5 | IC50 | 2 | — |