Target Details
| UniProt AC | O43613 |
|---|---|
| Gene Symbol | HCRTR1 |
| Protein Name | Orexin/Hypocretin receptor type 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 3,881
- Clinical molecules 0
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (3,881)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TZAQHYIVSIBZMW
|
9.0 | IC50 | 2 | — | |
VCZBQPUFKCYVDZ
|
9.0 | Ki | 2 | — | |
WRPGNWQVJUWOTB
|
9.0 | Ki | 2 | — | |
WWEKFLWFASRPJA
|
9.0 | IC50 | 2 | — | |
XVMJBFKNJYLIGG
|
9.0 | IC50 | 2 | — | |
YCPDCUAUNGQDQS
|
9.0 | IC50 | 2 | — | |
YMUFJVXLZBNCCA
|
9.0 | Ki | 2 | — | |
AEZZJXJIJFSUEM
|
9.0 | IC50 | 2 | — | |
HYBZWVLPALMACV
|
9.0 | Ki | 2 | — | |
IQBQPKYTEMWHQG
|
9.0 | IC50 | 2 | — | |
IWNMAIDPCKYHEC
|
9.0 | IC50 | 2 | — | |
XIBNNBMLUUIACY
|
9.0 | IC50 | 2 | — | |
ZKGLIXSQQKFLED
|
9.0 | IC50 | 2 | — | |
AHMDYOOHWSZVAL
|
8.9 | Ki | 2 | — | |
FRTWAZCPGVVGAL
|
8.9 | Ki | 2 | — | |
RDMQLFQIFXFJMN
|
8.9 | Ki | 2 | — | |
VENYONTWRDJMIS
|
8.9 | IC50 | 2 | — | |
WRTKUBDGKZTJTN
|
8.9 | IC50 | 2 | — | |
ZDVFZRUEEUXZRL
|
8.9 | IC50 | 2 | — | |
VCYRJXZNOOUBSE
|
8.9 | Ki | 2 | — | |
UJGSPBJSTPPWNS
|
8.9 | Ki | 2 | — | |
DSGAQPGARLXAPN
|
8.9 | Ki | 2 | — | |
NOGNYOCHJGNNCS
|
8.8 | IC50 | 2 | — | |
JYTNQNCOQXFQPK
|
8.8 | Ki | 2 | — | |
IRHPPLSFVLVHBZ
|
8.8 | IC50 | 2 | — | |
PETFZHTTWWEOOY
|
8.8 | Ki | 2 | — | |
DPEDZHZCLRBPSO
|
8.8 | IC50 | 2 | — | |
HWGBBJAHMAYQFQ
|
8.8 | Ki | 2 | — | |
PVUUFIVOJFEQPA
|
8.8 | Ki | 2 | — | |
SVSUWORSBYUYII
|
8.8 | IC50 | 2 | — | |
UCTMYARPCLQYDJ
|
8.8 | IC50 | 2 | — | |
HMLZGOXPNQUWLR
|
8.8 | IC50 | 2 | — | |
FASRRZAOIXPOCE
|
8.7 | IC50 | 2 | — | |
GOTIIFLZZULEEL
|
8.7 | Ki | 2 | — | |
HNNSGEZQVPZHPI
|
8.7 | IC50 | 2 | — | |
LPFZYIGBGPEIEZ
|
8.7 | IC50 | 2 | — | |
OAATXFVQEMAHDA
|
8.7 | Ki | 2 | — | |
SSVVKBOEKJMVND
|
8.7 | IC50 | 2 | — | |
AEIYXQGHBFFFPX
|
8.7 | IC50 | 2 | — | |
GESLELVSGPTNFL
|
8.7 | IC50 | 2 | — | |
YLBYPMTXVWAXOX
|
8.7 | IC50 | 2 | — | |
MPIPRURYZBEAQW
|
8.7 | Ki | 2 | — | |
AESOLJVLORXMKZ
|
8.7 | Ki | 2 | — | |
ALXXSSTULXRROK
|
8.7 | IC50 | 2 | — | |
APWITTXYMQNNTN
|
8.7 | IC50 | 2 | — | |
BHYJNXZXWCRENL
|
8.7 | IC50 | 2 | — | |
CGJIPORKYPTNBC
|
8.7 | IC50 | 2 | — | |
CKIBODIXGNACEX
|
8.7 | Ki | 2 | — | |
CYPZFHYWAMSWRL
|
8.7 | IC50 | 2 | — | |
DCMSTVVYTKCBDX
|
8.7 | IC50 | 2 | — |