Target Details
| UniProt AC | O43613 |
|---|---|
| Gene Symbol | HCRTR1 |
| Protein Name | Orexin/Hypocretin receptor type 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 3,881
- Clinical molecules 0
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (3,881)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QTGVVJKIDVNSKU
|
9.1 | IC50 | 2 | — | |
SUUDDUCMECPZLW
|
9.1 | IC50 | 2 | — | |
ZKDXPQCTBSYECW
|
9.1 | IC50 | 2 | — | |
ZSFKTFCHCZQVDT
|
9.1 | IC50 | 2 | — | |
HDXOKNFWVWBAOR
|
9.0 | Kd | 2 | — | |
ACKAOVNXPNOWIE
|
9.0 | IC50 | 2 | — | |
AWDZNHIULYTTNC
|
9.0 | IC50 | 2 | — | |
AZKADNWHMIVDCE
|
9.0 | IC50 | 2 | — | |
BJMYJAPKIHPIPW
|
9.0 | IC50 | 2 | — | |
BSPIQLLFYKKPND
|
9.0 | IC50 | 2 | — | |
BTNLZELUPKRKLO
|
9.0 | IC50 | 2 | — | |
CMHMTFXCDBXJMB
|
9.0 | Ki | 2 | — | |
CMSWWEXLVMHQNL
|
9.0 | IC50 | 2 | — | |
CNZCWXXEJIVJJI
|
9.0 | IC50 | 2 | — | |
CSNOPSKKXVIYCS
|
9.0 | IC50 | 2 | — | |
CZXWCWCRILWJKE
|
9.0 | IC50 | 2 | — | |
FPUDWXNHINXQHL
|
9.0 | Ki | 2 | — | |
HBIJQRRDMMOOSE
|
9.0 | IC50 | 2 | — | |
HFYYHVKYLPJNOE
|
9.0 | IC50 | 2 | — | |
HUPRZYCCDOZRQO
|
9.0 | IC50 | 2 | — | |
JHGRYXUHXJQVFP
|
9.0 | IC50 | 2 | — | |
JKTONSFRVQDZTK
|
9.0 | IC50 | 2 | — | |
JOAYSRXNJHJJBL
|
9.0 | IC50 | 2 | — | |
KANLBBSZECYCLU
|
9.0 | IC50 | 2 | — | |
KSJSBJPGMOQINA
|
9.0 | IC50 | 2 | — | |
LRBYYJMSSHIJKG
|
9.0 | IC50 | 2 | — | |
MCOBUUIPLMSSOE
|
9.0 | IC50 | 2 | — | |
MDIAYXGXQBIAME
|
9.0 | IC50 | 2 | — | |
MOXXGRCLAOBXLS
|
9.0 | IC50 | 2 | — | |
MPGPDRPDYBLHHF
|
9.0 | IC50 | 2 | — | |
NFAMQGWLSKBGPG
|
9.0 | IC50 | 2 | — | |
NIEKUZAHPSOMLB
|
9.0 | IC50 | 2 | — | |
NNEYHDHJHDRFBV
|
9.0 | IC50 | 2 | — | |
OBJHSZWESOSYIS
|
9.0 | IC50 | 2 | — | |
ONVKTAGSXCPXIK
|
9.0 | IC50 | 2 | — | |
ORXQOPADZCARMN
|
9.0 | IC50 | 2 | — | |
OZQQWERPXKWLAA
|
9.0 | IC50 | 2 | — | |
PGYQLCUKNOYWCZ
|
9.0 | IC50 | 2 | — | |
PLSLMYBUUIRIHB
|
9.0 | IC50 | 2 | — | |
PYSPVSXASXGIRN
|
9.0 | IC50 | 2 | — | |
PYTQJNRFZSSECU
|
9.0 | IC50 | 2 | — | |
QFDUIRFVMRTEFQ
|
9.0 | IC50 | 2 | — | |
QGLAATQFBFNUCL
|
9.0 | IC50 | 2 | — | |
RFRBKJBYJXZXKQ
|
9.0 | IC50 | 3 | — | |
RGQDQGMCUZKIIP
|
9.0 | IC50 | 2 | — | |
SABPYUNGMHYDLK
|
9.0 | IC50 | 2 | — | |
SDFNCQZAYMVNNG
|
9.0 | IC50 | 2 | — | |
SVWRBCQUGLPUCX
|
9.0 | IC50 | 2 | — | |
SWJLISCOLSUHGG
|
9.0 | Ki | 2 | — | |
SXDFZCLHFGCOFB
|
9.0 | IC50 | 2 | — |