Target Details
| UniProt AC | O43497 |
|---|---|
| Gene Symbol | CACNA1G |
| Protein Name | Voltage-dependent T-type calcium channel subunit alpha-1G |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) |
Summary
- Multi-target molecules 265
- Clinical molecules 1
- Avg pChEMBL 7.3
KEGG Pathways (8)
Associated Diseases (1)
Active Molecules (265)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LLVALEUPUXIQNY
|
6.6 | IC50 | 2 | — | |
SHBCBFDPLIFTBC
|
6.6 | IC50 | 3 | — | |
GLVAZBLDEWPYAU
|
6.6 | IC50 | 2 | — | |
JHTZHLHQRYYYJC
|
6.6 | IC50 | 3 | — | |
OWTDJGCKDWJAIU
|
6.6 | IC50 | 2 | — | |
LMXBXUWYKUDWME
|
6.6 | IC50 | 3 | — | |
QKTMLCGPKFUYDS
|
6.6 | IC50 | 2 | — | |
UYFGCFWWQASWNQ
|
6.6 | IC50 | 2 | — | |
UXVGOSYIXODHIO
|
6.6 | IC50 | 3 | — | |
JFGVQJFBQJWZAW
|
6.6 | IC50 | 3 | — | |
PYKGDXMPNNOJAK
|
6.6 | IC50 | 3 | — | |
QGMUDAKKGSLGLA
|
6.6 | IC50 | 3 | — | |
IQLMMMGWBQPWOW
|
6.5 | IC50 | 2 | — | |
JFGVQJFBQJWZAW
|
6.5 | IC50 | 3 | — | |
GEMLUIAYLYXCRN
|
6.5 | IC50 | 3 | — | |
YLBJFQXCNGOXMS
|
6.5 | IC50 | 3 | — | |
GYZMZXNNALBNTL
|
6.5 | IC50 | 3 | — | |
XWSPLWBSYSPPFJ
|
6.5 | IC50 | 3 | — | |
AKPBGOZQZZJVAV
|
6.5 | IC50 | 3 | — | |
FGOMAEMCCGRKRQ
|
6.5 | IC50 | 3 | — | |
WDGLTPTVGIOJHF
|
6.5 | IC50 | 2 | — | |
CKEKSOUQZDEDNJ
|
6.5 | IC50 | 2 | — | |
SBLBZIGASSBPMO
|
6.5 | IC50 | 3 | — | |
JZRTUPOQWXLSSB
|
6.4 | IC50 | 3 | — | |
PDUDKACBOWTICF
|
6.4 | IC50 | 2 | — | |
DXHGSDDDNQXAEJ
|
6.4 | IC50 | 26 | — | |
MGJWWKFNLMFMAB
|
6.4 | IC50 | 2 | — | |
MXPIHVJVTXGYGQ
|
6.4 | IC50 | 3 | — | |
KUOONLAXIFFQSP
|
6.4 | IC50 | 2 | — | |
IISKPGDTZKNEGX
|
6.4 | IC50 | 3 | — | |
JZRTUPOQWXLSSB
|
6.4 | IC50 | 3 | — | |
AZYQONGTQTXNKA
|
6.3 | IC50 | 3 | — | |
LAYLVIDKHAQDFA
|
6.3 | IC50 | 3 | — | |
LVGXCEUSAHWSLB
|
6.3 | IC50 | 2 | — | |
MLTMYDVQCHBUPB
|
6.3 | IC50 | 3 | — | |
UOXOWMNNZYBJHK
|
6.3 | IC50 | 3 | — | |
QZMUXWOFSPBIOL
|
6.3 | IC50 | 2 | — | |
GSMBBFLAEIUAQY
|
6.3 | IC50 | 3 | — | |
JIMHZFYOORSBOB
|
6.3 | IC50 | 2 | — | |
SMANXXCATUTDDT
|
6.3 | Kd | 25 | Yes | |
FMQVPNGZFBGFFN
|
6.3 | IC50 | 2 | — | |
QGXCVEORRPKPGU
|
6.2 | IC50 | 2 | — | |
YSJQTBCCKOJHFP
|
6.2 | IC50 | 3 | — | |
DVUQADUMMXGGPJ
|
6.2 | IC50 | 3 | — | |
GIBDJBDXOPLUGD
|
6.2 | IC50 | 3 | — | |
MULAMVHSOJFSOK
|
6.2 | IC50 | 2 | — | |
RLIKJYGXUGWLOZ
|
6.2 | IC50 | 3 | — | |
CWYZYWVFYWIMBI
|
6.2 | IC50 | 2 | — | |
NGUAIHUUBCVZQW
|
6.2 | IC50 | 2 | — | |
QHKJELCIBOZDRA
|
6.2 | IC50 | 2 | — |