Target Details
| UniProt AC | O43463 |
|---|---|
| Gene Symbol | SUV39H1 |
| Protein Name | Histone-lysine N-methyltransferase SUV39H1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00385 (Chromo) PF05033 (Pre-SET) PF00856 (SET) |
Summary
- Multi-target molecules 4
- Clinical molecules 1
- Avg pChEMBL 6.54
KEGG Pathways (2)
Active Molecules (4)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZRZWBWPDBOVIGQ
|
7.2 | IC50 | 4 | — | |
FIVPIPIDMRVLAY
|
6.6 | IC50 | 7 | Yes | |
PVVLIIZIQXDFSP
|
6.3 | IC50 | 2 | — | |
PZPPOCZWRGNKIR
|
6.1 | IC50 | 2 | — |