Target Details
| UniProt AC | O43353 |
|---|---|
| Gene Symbol | RIPK2 |
| Protein Name | Receptor-interacting serine/threonine-protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00619 (CARD) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 210
- Clinical molecules 19
- Avg pChEMBL 7.3
KEGG Pathways (5)
Active Molecules (210)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VKSOIYNNOFGGES
|
6.1 | IC50 | 3 | — | |
KTEIFNKAUNYNJU
|
6.0 | Kd | 114 | — | |
VKSOIYNNOFGGES
|
6.0 | IC50 | 2 | — | |
HXHAJRMTJXHJJZ
|
6.0 | Kd | 52 | Yes | |
YABJJWZLRMPFSI
|
6.0 | Kd | 34 | — | |
NHHQJBCNYHBUSI
|
6.0 | Kd | 220 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
LVXJQMNHJWSHET
|
6.0 | Kd | 7 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |