Target Details
| UniProt AC | O43353 |
|---|---|
| Gene Symbol | RIPK2 |
| Protein Name | Receptor-interacting serine/threonine-protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00619 (CARD) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 210
- Clinical molecules 19
- Avg pChEMBL 7.3
KEGG Pathways (5)
Active Molecules (210)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UIIXJLLQKFFGKU
|
7.4 | IC50 | 3 | — | |
SFZONKARGQSFPV
|
7.4 | IC50 | 2 | — | |
MOHYPRXHKRXDSE
|
7.4 | IC50 | 8 | — | |
XAVIPIHNPPAYAJ
|
7.4 | IC50 | 3 | — | |
SLEWGGZPOQNVSU
|
7.4 | Kd | 22 | — | |
IVRXNBXKWIJUQB
|
7.4 | IC50 | 10 | — | |
LPFWVDIFUFFKJU
|
7.3 | Kd | 9 | — | |
YFYPWCVYZUWOGM
|
7.3 | IC50 | 2 | — | |
WKHMETWKHWYTEE
|
7.3 | IC50 | 2 | — | |
WTNLXMJMLHJDKF
|
7.3 | IC50 | 3 | — | |
FJCDSQATIJKQKA
|
7.3 | IC50 | 5 | — | |
RVYNOQUUDOREOT
|
7.3 | IC50 | 2 | — | |
QRDCOOSKIFYKIQ
|
7.2 | Kd | 8 | — | |
XYFPWWZEPKGCCK
|
7.2 | Kd | 34 | — | |
JOJOVBICKPOJFI
|
7.2 | IC50 | 3 | — | |
BRZGXSNAXRPPFI
|
7.2 | IC50 | 2 | — | |
BGIYKDUASORTBB
|
7.2 | IC50 | 6 | — | |
YULUHUJTIHWRMI
|
7.2 | Kd | 4 | — | |
FAXUBOMVBMGLNX
|
7.2 | IC50 | 2 | — | |
MCKKWYKONXTPFI
|
7.1 | IC50 | 3 | — | |
MLDQJTXFUGDVEO
|
7.1 | IC50 | 85 | Yes | |
BFSMGDJOXZAERB
|
7.1 | IC50 | 33 | — | |
MFAQYJIYDMLAIM
|
7.1 | Kd | 130 | Yes | |
WKTLXYXOPICQKS
|
7.1 | IC50 | 2 | — | |
XASOHFCUIQARJT
|
7.1 | IC50 | 4 | — | |
FQUBTLMSWPIBBP
|
7.1 | Kd | 4 | — | |
HDMLUZMVBVBTJX
|
7.1 | IC50 | 2 | — | |
UVHMCYBDLLCIAP
|
7.1 | IC50 | 2 | — | |
AHESYZXOYPHUOT
|
7.1 | Kd | 4 | — | |
CIKRVGZNQZNXMQ
|
7.0 | IC50 | 2 | — | |
VYPGLYMWNDRFGZ
|
7.0 | Kd | 12 | — | |
ORTYQHFTTCRJIP
|
7.0 | IC50 | 2 | — | |
BLWQIEISIMYCHD
|
7.0 | Kd | 4 | — | |
UMLPCOVOJFEKRE
|
7.0 | IC50 | 2 | — | |
UQRCJCNVNUFYDX
|
7.0 | Kd | 27 | — | |
XXJWYDDUDKYVKI
|
7.0 | Kd | 52 | — | |
BHUXVRVMMYAXKN
|
7.0 | IC50 | 3 | — | |
RIEGJNXDHULIKM
|
7.0 | IC50 | 3 | — | |
UPGITVUUJFWGDH
|
7.0 | IC50 | 2 | — | |
CKZNIIZTVZQXIP
|
7.0 | IC50 | 2 | — | |
AUOSKLDNVNGKRR
|
7.0 | Kd | 6 | — | |
RYKSGWSKILPDDY
|
7.0 | IC50 | 4 | — | |
XSHQBIXMLULFEV
|
6.9 | IC50 | 13 | — | |
QKIQUHJMKMTYPI
|
6.9 | IC50 | 2 | — | |
YLQIGGIFOQEJNU
|
6.9 | IC50 | 2 | — | |
GDQXJQSQYMMKRA
|
6.9 | IC50 | 15 | — | |
MJZHYLCYHDBDFA
|
6.9 | IC50 | 2 | — | |
WUEJFDOJIBRVBJ
|
6.9 | IC50 | 3 | — | |
XKNAGLMNQADBQE
|
6.8 | IC50 | 2 | — | |
PDZAPYOZOLWESW
|
6.8 | IC50 | 4 | — |