Target Details
| UniProt AC | O43318 |
|---|---|
| Gene Symbol | MAP3K7 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 178
- Clinical molecules 12
- Avg pChEMBL 6.96
KEGG Pathways (29)
- AMPK signaling pathway
- Adherens junction
- Alcoholic liver disease
- Autophagy - animal
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Fluid shear stress and atherosclerosis
- Hepatitis B
- Herpes simplex virus 1 infection
- Human immunodeficiency virus 1 infection
- IL-17 signaling pathway
- Leishmaniasis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- Pathogenic Escherichia coli infection
- RIG-I-like receptor signaling pathway
- Salmonella infection
- Shigellosis
- T cell receptor signaling pathway
- TNF signaling pathway
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Wnt signaling pathway
- Yersinia infection
Associated Diseases (2)
Active Molecules (178)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SPEMUMBPRQTTAA
|
6.7 | IC50 | 2 | — | |
PPCIDOUXWYIBPO
|
6.7 | IC50 | 6 | — | |
FJPOGNAHCZFDQR
|
6.6 | IC50 | 2 | — | |
ONRYANARCHPXRQ
|
6.6 | IC50 | 2 | — | |
SMIIJPDEPOIIHO
|
6.6 | IC50 | 2 | — | |
CJQGLUJHMXCLQY
|
6.6 | IC50 | 11 | — | |
NANIKNNTSLTWED
|
6.6 | IC50 | 2 | — | |
WZBIRANKKAOEQU
|
6.6 | IC50 | 2 | — | |
KJHFJTDIYVBYIY
|
6.5 | IC50 | 2 | — | |
PONZXJHPMSOTCH
|
6.5 | IC50 | 2 | — | |
OLKMNKWCYPTDSI
|
6.5 | IC50 | 2 | — | |
JNOGMCOTCINPDR
|
6.5 | IC50 | 2 | — | |
QMKZTPJYKZRXJU
|
6.5 | IC50 | 2 | — | |
UEJPPFOPQURDKT
|
6.5 | IC50 | 2 | — | |
WPLBZSRCAZTCEF
|
6.5 | IC50 | 2 | — | |
OQDJNLKOMYTWEB
|
6.5 | IC50 | 2 | — | |
SUSVWEQZHZXFBT
|
6.5 | IC50 | 2 | — | |
DSQSRIOQMWVLNQ
|
6.5 | IC50 | 2 | — | |
ASMLDRAEBPYENO
|
6.5 | IC50 | 10 | — | |
FCNPQYHKUYSELK
|
6.4 | IC50 | 8 | — | |
PXVURKNFXLGXEF
|
6.4 | IC50 | 2 | — | |
QZUXSJFGHNXNFE
|
6.4 | IC50 | 2 | — | |
YIGLAOIVUJQLRW
|
6.4 | IC50 | 2 | — | |
NTJCHTSHOGWLTQ
|
6.4 | IC50 | 2 | — | |
PPDQFCISGDOHIO
|
6.4 | IC50 | 2 | — | |
VYOVIFUEUXGCRT
|
6.4 | IC50 | 2 | — | |
KEAPLOABAMRRFQ
|
6.4 | IC50 | 2 | — | |
HNRZIHVCJQLPHG
|
6.4 | IC50 | 2 | — | |
QTEKWFKGOIRYGW
|
6.4 | IC50 | 2 | — | |
OUAQOOWAHVGVHU
|
6.4 | IC50 | 2 | — | |
SNKIPAIHEQSWBK
|
6.3 | IC50 | 2 | — | |
ZJOCDAGVCZOCSS
|
6.3 | IC50 | 2 | — | |
NOINHGBAXKOKQW
|
6.3 | IC50 | 2 | — | |
NXNILAJGBIVOOD
|
6.3 | IC50 | 2 | — | |
OFGWSAWNQPAURN
|
6.3 | IC50 | 2 | — | |
MBDDGSKUZPVINA
|
6.3 | IC50 | 2 | — | |
WPXVVAWAHQHJPF
|
6.3 | IC50 | 41 | — | |
YABJJWZLRMPFSI
|
6.3 | Kd | 34 | — | |
UEJPPFOPQURDKT
|
6.3 | IC50 | 2 | — | |
XESCBULBTJHJDG
|
6.3 | IC50 | 2 | — | |
CXQHYVUVSFXTMY
|
6.3 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.3 | Kd | 149 | — | |
DNUSNALEWBPUMU
|
6.2 | IC50 | 2 | — | |
RCXJDSKUXDREIO
|
6.2 | IC50 | 2 | — | |
XCKISTZRDFIEIS
|
6.2 | IC50 | 2 | — | |
ZINYHYQBLSXMQW
|
6.2 | IC50 | 2 | — | |
BKLVJHYYETWJAN
|
6.2 | IC50 | 2 | — | |
FQVJFULIWJSXIM
|
6.2 | IC50 | 2 | — | |
PIQCTGMSNWUMAF
|
6.2 | Kd | 137 | Yes | |
BPNUQXPIQBZCMR
|
6.2 | Kd | 83 | Yes |