Target Details
| UniProt AC | O43318 |
|---|---|
| Gene Symbol | MAP3K7 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 178
- Clinical molecules 12
- Avg pChEMBL 6.96
KEGG Pathways (29)
- AMPK signaling pathway
- Adherens junction
- Alcoholic liver disease
- Autophagy - animal
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Fluid shear stress and atherosclerosis
- Hepatitis B
- Herpes simplex virus 1 infection
- Human immunodeficiency virus 1 infection
- IL-17 signaling pathway
- Leishmaniasis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- Pathogenic Escherichia coli infection
- RIG-I-like receptor signaling pathway
- Salmonella infection
- Shigellosis
- T cell receptor signaling pathway
- TNF signaling pathway
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Wnt signaling pathway
- Yersinia infection
Associated Diseases (2)
Active Molecules (178)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ASCPSRDSSMPJDW
|
7.3 | IC50 | 3 | — | |
IBYHNCOWDYTTRQ
|
7.3 | IC50 | 2 | — | |
NHHQJBCNYHBUSI
|
7.3 | Kd | 220 | — | |
YHVHYWYQEFELOW
|
7.3 | IC50 | 44 | — | |
KFTLSWHJVMUFGV
|
7.3 | IC50 | 2 | — | |
RUNVBUSNWGRNAS
|
7.3 | IC50 | 2 | — | |
KYNJAMYDYPTYDZ
|
7.2 | IC50 | 2 | — | |
ZWXIOQDBSVHEGC
|
7.2 | IC50 | 2 | — | |
OSVUGUHRKMMBSE
|
7.2 | Kd | 170 | — | |
BNRXMSGHPVYSDK
|
7.2 | IC50 | 24 | — | |
ANCZNPGQXFLAIW
|
7.2 | IC50 | 3 | — | |
LHDKPFSHXFFALR
|
7.2 | IC50 | 7 | — | |
HKSZLNNOFSGOKW
|
7.2 | IC50 | 408 | — | |
LSSSBVSRWFCJKB
|
7.1 | IC50 | 2 | — | |
XLFJEGWLJGWRSM
|
7.1 | IC50 | 4 | — | |
VGAICDJDNKCITB
|
7.1 | IC50 | 2 | — | |
FKDNUEBNRIFBDZ
|
7.1 | IC50 | 3 | — | |
OACJMCGKLHFOLN
|
7.0 | IC50 | 2 | — | |
WINHZLLDWRZWRT
|
7.0 | Kd | 201 | Yes | |
WANRGEOLLIFNBS
|
7.0 | Kd | 4 | — | |
OMSUAZHPXSYOQO
|
7.0 | IC50 | 2 | — | |
CTNPALGJUAXMMC
|
7.0 | Kd | 151 | — | |
MIWFIZLZRBKGQU
|
7.0 | IC50 | 2 | — | |
UBPYILGKFZZVDX
|
7.0 | Kd | 130 | Yes | |
XGQCOOMJAUFAOT
|
7.0 | IC50 | 2 | — | |
ZFLJQOGIHBIDNZ
|
7.0 | IC50 | 2 | — | |
LTQRMOSYFBRQRH
|
6.9 | IC50 | 2 | — | |
RPDGGTQIKZCYAP
|
6.9 | IC50 | 3 | — | |
UUSDUSGMWIXJOT
|
6.9 | IC50 | 2 | — | |
AMHWQBGAKJESFB
|
6.9 | IC50 | 4 | — | |
BMGQWWVMWDBQGC
|
6.9 | Kd | 147 | Yes | |
JXNXZCJQWOEXJV
|
6.9 | IC50 | 2 | — | |
UUTHPYJPFVUVPN
|
6.9 | Ki | 3 | — | |
IHXGKMUEVBBWBZ
|
6.9 | IC50 | 2 | — | |
SMPGEBOIKULBCT
|
6.8 | IC50 | 15 | — | |
MVCOAUNKQVWQHZ
|
6.8 | Kd | 54 | Yes | |
PCFQERXLBAHWRY
|
6.8 | IC50 | 4 | — | |
BUZQLQAPFVMMQY
|
6.8 | IC50 | 2 | — | |
QQWUGDVOUVUTOY
|
6.8 | Kd | 231 | Yes | |
JIOOBLLPEPCAAJ
|
6.8 | IC50 | 4 | — | |
PCGJEVAVUOYIQB
|
6.8 | IC50 | 2 | — | |
SPEMUMBPRQTTAA
|
6.8 | IC50 | 2 | — | |
UPJJRELFFCGJGA
|
6.8 | IC50 | 2 | — | |
ZDIREJTXQKRZCD
|
6.8 | IC50 | 2 | — | |
NTUWMPKGQOZJLQ
|
6.8 | IC50 | 2 | — | |
OUCUNVKXSOPBBS
|
6.7 | IC50 | 4 | — | |
YYTVWIMHEXZBKS
|
6.7 | IC50 | 2 | — | |
FCYFQTBWJKSDFR
|
6.7 | IC50 | 2 | — | |
YSMQCLKSRAHMMV
|
6.7 | IC50 | 2 | — | |
LQSGDXCDNZWTJN
|
6.7 | IC50 | 17 | — |