Target Details
| UniProt AC | O43318 |
|---|---|
| Gene Symbol | MAP3K7 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 178
- Clinical molecules 12
- Avg pChEMBL 6.96
KEGG Pathways (29)
- AMPK signaling pathway
- Adherens junction
- Alcoholic liver disease
- Autophagy - animal
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Fluid shear stress and atherosclerosis
- Hepatitis B
- Herpes simplex virus 1 infection
- Human immunodeficiency virus 1 infection
- IL-17 signaling pathway
- Leishmaniasis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- Pathogenic Escherichia coli infection
- RIG-I-like receptor signaling pathway
- Salmonella infection
- Shigellosis
- T cell receptor signaling pathway
- TNF signaling pathway
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Wnt signaling pathway
- Yersinia infection
Associated Diseases (2)
Active Molecules (178)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ODPGGGTTYSGTGO
|
8.8 | Kd | 153 | — | |
MENPTCWEPFMOHL
|
8.8 | IC50 | 3 | — | |
QEAYKBGEHPZBIL
|
8.7 | IC50 | 2 | — | |
USMAPSJMQVFIAW
|
8.6 | IC50 | 2 | — | |
ORBLOJJZDLUQDF
|
8.6 | IC50 | 4 | — | |
UIARLYUEJFELEN
|
8.5 | Kd | 289 | Yes | |
RNDSPZADISTGBT
|
8.5 | IC50 | 2 | — | |
NGMAFXVXLJNKNC
|
8.5 | IC50 | 3 | — | |
XZXHXSATPCNXJR
|
8.4 | Kd | 165 | Yes | |
JURMELNKITYBRM
|
8.4 | IC50 | 2 | — | |
YQZZHUQLRWPXNZ
|
8.4 | IC50 | 2 | — | |
WUOCHAVLTKNGCC
|
8.3 | IC50 | 2 | — | |
JTCXCSWNNQIPRO
|
8.3 | IC50 | 2 | — | |
FVFLNMVKWNRXOS
|
8.3 | IC50 | 2 | — | |
WVXNSAVVKYZVOE
|
8.2 | IC50 | 92 | — | |
XDCWLOMVUOZXFY
|
8.2 | IC50 | 2 | — | |
JDBLJGQEXWERKN
|
8.2 | IC50 | 3 | — | |
ZQACLJMUNJMDKP
|
8.2 | IC50 | 2 | — | |
GUBJNPWVIUFSTR
|
8.1 | Kd | 103 | — | |
QXQGHCJUTRTRLJ
|
8.1 | IC50 | 2 | — | |
IWIYCPMVAVQALP
|
8.1 | IC50 | 2 | — | |
VZWXALUQDOYOJQ
|
8.1 | IC50 | 2 | — | |
NEQZWEXWOFPKOT
|
8.1 | IC50 | 9 | — | |
CGZANCKEFIHBJE
|
8.0 | IC50 | 2 | — | |
SLKSOMMHRLEOCJ
|
8.0 | IC50 | 2 | — | |
UNYPOOKIBOGJII
|
7.9 | IC50 | 2 | — | |
WFHQLAWBICSWPO
|
7.9 | IC50 | 4 | — | |
OIZYRHLPFJOIQM
|
7.9 | IC50 | 2 | — | |
DGUFRRJUHIZTQE
|
7.8 | Ki | 3 | — | |
IIBQLYSZHMEQIH
|
7.8 | IC50 | 2 | — | |
CQMWAJCVQYHQCJ
|
7.8 | IC50 | 2 | — | |
FLZAOAIEJUXTAH
|
7.8 | IC50 | 2 | — | |
MJJJFOLDERHCND
|
7.7 | IC50 | 2 | — | |
PZPZZBSXXDLNMN
|
7.7 | IC50 | 2 | — | |
IXXBWYJJOYSCNJ
|
7.6 | IC50 | 2 | — | |
QJGDGWJGAAATCO
|
7.6 | IC50 | 2 | — | |
ZOGZUMFMIBABFJ
|
7.6 | IC50 | 2 | — | |
VLSKNLVBBCEHSR
|
7.6 | IC50 | 2 | — | |
QPKFIZDVDMZSPR
|
7.5 | Ki | 3 | — | |
HREDYOVSBYDONU
|
7.5 | IC50 | 2 | — | |
BKXGJUGZEFIAJO
|
7.5 | IC50 | 2 | — | |
SSNQAUBBJYCSMY
|
7.5 | IC50 | 5 | — | |
QWDMOLLUOYFWOV
|
7.4 | IC50 | 3 | — | |
YYLKKYCXAOBSRM
|
7.4 | Kd | 191 | — | |
LEVZCGPPIDIGHW
|
7.4 | IC50 | 2 | — | |
HUFPFCSZVXOFRZ
|
7.4 | IC50 | 2 | — | |
RQFOIAOPEILIMX
|
7.4 | IC50 | 2 | — | |
RWNAOXLCVXJMGM
|
7.4 | IC50 | 5 | — | |
UMBFDGUGXMOMHX
|
7.4 | IC50 | 12 | — | |
NXSJMRCTGYTSTK
|
7.4 | Kd | 200 | — |