Target Details
| UniProt AC | O43293 |
|---|---|
| Gene Symbol | DAPK3 |
| Protein Name | Death-associated protein kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 258
- Clinical molecules 20
- Avg pChEMBL 6.82
KEGG Pathways (3)
Active Molecules (258)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TWZVBMXTDSNZLS
|
6.3 | Ki | 7 | — | |
UEZPPFDNXOFISI
|
6.3 | Ki | 6 | — | |
YOVNFNXUCOWYSG
|
6.3 | Ki | 33 | Yes | |
ZRQXCQXWTLVASO
|
6.3 | Ki | 36 | — | |
XKQNBVAZAFAZFL
|
6.3 | IC50 | 6 | — | |
KGPGFQWBCSZGEL
|
6.2 | Kd | 59 | Yes | |
WPPGBVWZGMDXKF
|
6.2 | IC50 | 5 | — | |
GUMBHNMWKMFKRT
|
6.2 | Ki | 23 | — | |
HSKVRPZJBMXFDX
|
6.2 | Ki | 20 | — | |
IABDKYMGRMDGMM
|
6.2 | Ki | 10 | — | |
IMMZLRQJNZSTTE
|
6.2 | Ki | 15 | — | |
ISEDKXOMRIKZPK
|
6.2 | Ki | 13 | — | |
JPOSFPUHBHRUAX
|
6.2 | Ki | 40 | Yes | |
LHQWPYOYDRVMFI
|
6.2 | Ki | 21 | — | |
NRZYTPAJGVTKIM
|
6.2 | Ki | 38 | — | |
QZIVKBVZTKZHCY
|
6.2 | Ki | 2 | — | |
WAKGEHXTOOFEAE
|
6.2 | Ki | 27 | — | |
XJJYJNMNYDNXNO
|
6.2 | Ki | 23 | — | |
ZKZXNDJNWUTGDK
|
6.2 | Ki | 14 | — | |
QVJYGMLAIWRCFT
|
6.2 | IC50 | 5 | — | |
ACLLLJSNOCYQOJ
|
6.1 | IC50 | 8 | — | |
AEYLJTAIDDIOBA
|
6.1 | Ki | 53 | — | |
AWJPVXSHMIELNJ
|
6.1 | Ki | 23 | — | |
FPQHXFMYXQZPSV
|
6.1 | Ki | 23 | — | |
GSXRCPJTNIGKSZ
|
6.1 | Ki | 43 | — | |
KDJGCVHPUMHUOL
|
6.1 | Ki | 11 | — | |
KNARVZUUCLIBGV
|
6.1 | Ki | 33 | — | |
KYACBMRLQMEIAI
|
6.1 | Ki | 30 | — | |
LUPCHAFIKZSOOK
|
6.1 | Ki | 15 | — | |
QONPPIZSNSSCSK
|
6.1 | Ki | 45 | Yes | |
SFPWNTQWFFNJIH
|
6.1 | Ki | 48 | — | |
UIRCQOKSJDLYBB
|
6.1 | Ki | 50 | — | |
WZBMMJKAHHOXRG
|
6.1 | Ki | 16 | — | |
XKFTZKGMDDZMJI
|
6.1 | Ki | 56 | — | |
YWITWZUKNXWOSD
|
6.1 | Ki | 10 | — | |
ZTUKHYNMEWPBNZ
|
6.1 | Ki | 6 | — | |
TUVCWJQQGGETHL
|
6.1 | Kd | 22 | — | |
NXWXUDHOUKWAQU
|
6.1 | Kd | 16 | — | |
BZFGDXJGWSIYQP
|
6.0 | Ki | 9 | — | |
CPGKMMMSMJKHDL
|
6.0 | Ki | 16 | — | |
DZGATJHVQUFYSK
|
6.0 | Ki | 12 | — | |
FLHJZUQGFPJXRD
|
6.0 | Ki | 12 | — | |
GQHMZZXJWGPHDA
|
6.0 | Ki | 20 | — | |
IJNGXROUMFEKDB
|
6.0 | Ki | 39 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
LRINYHMQZRENCY
|
6.0 | Ki | 29 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MHCPAORAYMTGCZ
|
6.0 | Ki | 37 | — | |
MZDKLVOWGIOKTN
|
6.0 | Ki | 80 | — |