Target Details
| UniProt AC | O43293 |
|---|---|
| Gene Symbol | DAPK3 |
| Protein Name | Death-associated protein kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 258
- Clinical molecules 20
- Avg pChEMBL 6.82
KEGG Pathways (3)
Active Molecules (258)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VGURQCQNQDZAOF
|
6.6 | Ki | 6 | — | |
VXYDJXMHISGSDA
|
6.6 | Ki | 59 | — | |
WKWGFJFNCXAUEX
|
6.6 | Ki | 14 | Yes | |
XUGXUDSTKPTWNB
|
6.6 | Ki | 10 | — | |
YKYRQCWLYUTVIE
|
6.6 | Ki | 16 | — | |
ZGDYBJXDIXVTLV
|
6.6 | Ki | 54 | — | |
LOONVQWRKJLEEG
|
6.6 | IC50 | 8 | — | |
NASYEGAVCTZSDO
|
6.6 | Kd | 5 | — | |
YYLKKYCXAOBSRM
|
6.5 | Kd | 191 | — | |
ZUKXESAZGMJHLJ
|
6.5 | IC50 | 4 | — | |
CRKQBJZCCHKEGI
|
6.5 | Ki | 20 | — | |
DRTDDTWOOFJKOH
|
6.5 | Ki | 2 | — | |
GQLWKGVBOIYMTN
|
6.5 | Ki | 35 | — | |
GVMDVMPNOAVKJR
|
6.5 | Ki | 26 | Yes | |
KTWBYGUSEYSRND
|
6.5 | Ki | 28 | — | |
OUJZYQBEFNDJQN
|
6.5 | Ki | 71 | — | |
PJUVRETYCLPAFV
|
6.5 | Ki | 20 | — | |
QMMMGQKKOKYDMN
|
6.5 | Ki | 5 | — | |
UMYBAQLXZPEUQW
|
6.5 | Ki | 15 | — | |
UQFRSHRWRKYNDE
|
6.5 | Ki | 17 | Yes | |
VIJBEUTVNBPGIU
|
6.5 | Ki | 19 | — | |
VTQQYBGURNVVFE
|
6.5 | Ki | 17 | — | |
YGKFZWJWKPZPQM
|
6.5 | Ki | 13 | — | |
ZVWRFVCNQOECJS
|
6.5 | Ki | 71 | — | |
KOZFSFOOLUUIGY
|
6.4 | IC50 | 26 | — | |
CLRFYTGANQZOBS
|
6.4 | Ki | 41 | — | |
DZIPQNPWTUXXSJ
|
6.4 | Ki | 18 | — | |
GJOXRIYWDHESDF
|
6.4 | Ki | 27 | — | |
HHSVICUMCOBRPT
|
6.4 | Ki | 33 | — | |
IUEBPIPDFMCSTP
|
6.4 | Ki | 29 | — | |
OEKYVFZKBRIDJO
|
6.4 | Ki | 12 | — | |
QAJPIJHWTGPUNZ
|
6.4 | Ki | 37 | — | |
QCOULMVHIHJKFY
|
6.4 | Ki | 14 | — | |
QQWUGDVOUVUTOY
|
6.4 | Ki | 231 | Yes | |
RKUKAACYUCUJEE
|
6.4 | Ki | 58 | — | |
UJBJWYNPUOLFIZ
|
6.4 | Ki | 49 | — | |
VSVKFEMFAYXZKR
|
6.4 | Ki | 14 | Yes | |
KRIUNPBAQZGFQA
|
6.4 | Kd | 76 | — | |
LIMMMAWLSIHXGX
|
6.3 | IC50 | 5 | — | |
VVFCWFGNLTVHBL
|
6.3 | IC50 | 5 | — | |
NHDDTLMPCVOXFH
|
6.3 | IC50 | 16 | Yes | |
CLEGDJQQHUTCOW
|
6.3 | Ki | 43 | — | |
DPEXRCOBPACFOO
|
6.3 | Ki | 36 | — | |
FSWFKKQQSQHIRZ
|
6.3 | Ki | 10 | — | |
GQHSVFWCNBWKGM
|
6.3 | Ki | 3 | — | |
JJJSCYSPSKBQAX
|
6.3 | Ki | 34 | — | |
KXPWWMPXNUOYOH
|
6.3 | Ki | 24 | — | |
NLUPJKQOKWBWFC
|
6.3 | Ki | 69 | — | |
QGOIQRQXIWSNJF
|
6.3 | Ki | 6 | — | |
QLWUDWMYFSWGHK
|
6.3 | Ki | 22 | — |