Target Details
| UniProt AC | O43293 |
|---|---|
| Gene Symbol | DAPK3 |
| Protein Name | Death-associated protein kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 258
- Clinical molecules 20
- Avg pChEMBL 6.82
KEGG Pathways (3)
Active Molecules (258)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.0 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
9.0 | Kd | 213 | — | |
VNDWQCSOSCCWIP
|
9.0 | Ki | 39 | Yes | |
JOOXLOJCABQBSG
|
8.9 | Kd | 139 | — | |
HKSZLNNOFSGOKW
|
8.7 | Ki | 118 | — | |
JAMDNXUAYUHJLJ
|
8.6 | Ki | 40 | — | |
UMTWTCVTRDYHQQ
|
8.4 | Ki | 56 | — | |
NWMPVMMGSHXANZ
|
8.3 | Ki | 58 | — | |
ZKLJKKASNXVQBZ
|
8.3 | Ki | 27 | — | |
PNKALLUVKOKYHZ
|
8.1 | Ki | 32 | — | |
SDBOIBYRBWPIEL
|
8.1 | Ki | 31 | — | |
UDFDIIVNIYWXDM
|
8.1 | Ki | 74 | — | |
CYLGCMABIBXHIQ
|
7.9 | Ki | 16 | — | |
KHGPYYFCIAISBU
|
7.9 | Ki | 31 | — | |
PLHUMPJXRHMFFR
|
7.9 | Ki | 28 | — | |
CLYMONPGUOMIQL
|
7.9 | Kd | 3 | — | |
NHHQJBCNYHBUSI
|
7.9 | Kd | 220 | — | |
CKVWQORGCCEYHS
|
7.8 | Ki | 50 | — | |
GHMRUNOHAHJNNA
|
7.8 | Ki | 29 | — | |
JJTYLBBKGQOISV
|
7.8 | Ki | 15 | — | |
JOIUJUJSHIHBDT
|
7.8 | Ki | 18 | — | |
UYGYYOIUVFMGKQ
|
7.8 | Ki | 30 | — | |
MUOKSQABCJCOPU
|
7.8 | IC50 | 36 | — | |
BLQYVHBZHAISJM
|
7.7 | Ki | 54 | — | |
BSFNGHCTZDCQBF
|
7.7 | Ki | 93 | — | |
RJZDECGDCKOHBV
|
7.7 | Ki | 70 | — | |
RKKIDHHGKNGTQI
|
7.7 | Ki | 28 | — | |
WYOMXSAYYXBPMN
|
7.7 | Ki | 24 | — | |
WINHZLLDWRZWRT
|
7.7 | Kd | 201 | Yes | |
FQEODTMNWMDUMD
|
7.6 | Ki | 25 | — | |
HOYRWTWZUFFACV
|
7.6 | Ki | 28 | — | |
OSVUGUHRKMMBSE
|
7.6 | Kd | 170 | — | |
OWFLADWRSCINST
|
7.6 | Ki | 30 | — | |
SQXSMLLCDWJNAC
|
7.6 | Ki | 20 | — | |
XXSPHNFKLDJDAK
|
7.6 | Ki | 26 | — | |
HNODKCFEFLQKBO
|
7.5 | Ki | 6 | — | |
AOBLBPWPSKBHSI
|
7.5 | Ki | 55 | — | |
BGYVWFZMYBWCNY
|
7.5 | Ki | 30 | — | |
JXMYIDZREHNPDO
|
7.5 | Ki | 19 | — | |
MVJMMLFMPWITEJ
|
7.5 | Ki | 110 | — | |
VNGYQBMDQMDALH
|
7.5 | Ki | 25 | — | |
ZGZVRPRSFXRGCF
|
7.5 | Ki | 76 | — | |
ACSYKUPGCXYRRO
|
7.4 | Ki | 26 | — | |
HMKKDSBJGMESJD
|
7.4 | Ki | 10 | — | |
LACOMQAWPSFXQC
|
7.4 | Ki | 27 | — | |
NKGLJTITEFZKAN
|
7.4 | Ki | 35 | — | |
RWKDVIAVTRRJIR
|
7.4 | Ki | 23 | — | |
XPHWIERLJBFPFV
|
7.4 | Ki | 69 | — | |
ZPVLRSVLOWVDJC
|
7.4 | Ki | 14 | — | |
MFAQYJIYDMLAIM
|
7.4 | Kd | 130 | Yes |