Target Details
| UniProt AC | O43283 |
|---|---|
| Gene Symbol | MAP3K13 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 13 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 234
- Clinical molecules 8
- Avg pChEMBL 7.04
KEGG Pathways (1)
Active Molecules (234)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XYPSLUORQTXKII
|
6.3 | IC50 | 2 | — | |
KTICSPFVRMPOOD
|
6.3 | IC50 | 2 | — | |
YYLKKYCXAOBSRM
|
6.3 | Kd | 191 | — | |
CTNPALGJUAXMMC
|
6.3 | Kd | 151 | — | |
JPHUVBYQFLACGA
|
6.3 | IC50 | 2 | — | |
IPSIEHCTZGXLQW
|
6.2 | IC50 | 2 | — | |
JOOXLOJCABQBSG
|
6.2 | Kd | 139 | — | |
MHXWDVVRMXHYCD
|
6.2 | IC50 | 2 | — | |
IUHHKZYWPMOFAH
|
6.2 | IC50 | 2 | — | |
VJVIBFXROVNGMC
|
6.2 | IC50 | 2 | — | |
HLLYYRUWCUOBIF
|
6.2 | IC50 | 2 | — | |
HQZNAKDFOFNZRM
|
6.2 | IC50 | 2 | — | |
NPXKKYGDGPWDJG
|
6.2 | Kd | 2 | — | |
FOOHADSOTCVGKR
|
6.2 | IC50 | 2 | — | |
UEFDQVCCIABIGM
|
6.2 | IC50 | 2 | — | |
FZOXXDKWCWCPNU
|
6.2 | Kd | 2 | — | |
RVEPUEJNEZOKJM
|
6.2 | IC50 | 2 | — | |
DQMABCFMEBYHLF
|
6.2 | IC50 | 2 | — | |
JWNPDZNEKVCWMY
|
6.1 | Kd | 57 | Yes | |
ODPGGGTTYSGTGO
|
6.1 | Kd | 153 | — | |
YGSNUGAPYIPPAS
|
6.1 | IC50 | 2 | — | |
GNWLHTMNFDUEGD
|
6.1 | IC50 | 2 | — | |
JVLUYMQQLZKLSR
|
6.1 | IC50 | 2 | — | |
ZZVBIQXZAHZKGS
|
6.1 | IC50 | 2 | — | |
FAFMKRLHLJWOJO
|
6.1 | IC50 | 2 | — | |
RULZPIBUCBDGRW
|
6.1 | IC50 | 2 | — | |
UMIKNAVKPZPHFL
|
6.1 | Kd | 2 | — | |
IMJGAPDZBWUOKM
|
6.1 | IC50 | 2 | — | |
QLRTZMSAJQFZOS
|
6.0 | IC50 | 2 | — | |
QIZJZGQPQPHFPE
|
6.0 | IC50 | 2 | — | |
IFJRORWVQKJIQH
|
6.0 | IC50 | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |