Target Details
| UniProt AC | O43283 |
|---|---|
| Gene Symbol | MAP3K13 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 13 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 234
- Clinical molecules 8
- Avg pChEMBL 7.04
KEGG Pathways (1)
Active Molecules (234)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PKYXUUGDLNWHBZ
|
6.7 | Kd | 2 | — | |
JCDUHLOBPFQKTC
|
6.7 | IC50 | 2 | — | |
WVSYEVKDFSRHMH
|
6.7 | IC50 | 2 | — | |
AKKHHVJIISFQCL
|
6.7 | IC50 | 2 | — | |
ARXOCNZUYXHLEU
|
6.7 | IC50 | 2 | — | |
GUBJNPWVIUFSTR
|
6.7 | Kd | 103 | — | |
HKSZLNNOFSGOKW
|
6.7 | Kd | 408 | — | |
HOZQTQHWMQJEHD
|
6.7 | IC50 | 2 | — | |
YQDLJHIIPMOELB
|
6.7 | IC50 | 2 | — | |
FHYMWFXNNDZTOE
|
6.6 | IC50 | 2 | — | |
KTEIFNKAUNYNJU
|
6.6 | Kd | 114 | — | |
MHOZTJUZLOQMBX
|
6.6 | Kd | 2 | — | |
MKBRJNKXYINGBL
|
6.6 | Kd | 2 | — | |
XOFDSSNUFUJXNW
|
6.6 | Kd | 2 | — | |
LNGJQTNUWUUKKY
|
6.6 | IC50 | 2 | — | |
FQRCKINZIWCFBW
|
6.6 | IC50 | 2 | — | |
RBMVDIMGHJCANE
|
6.6 | Kd | 2 | — | |
VWIJCPJOMFBEQC
|
6.6 | IC50 | 2 | — | |
YGSNUGAPYIPPAS
|
6.6 | IC50 | 2 | — | |
XGFVOKJJQCQLJX
|
6.6 | IC50 | 2 | — | |
FSTMHVBLNXUGCA
|
6.6 | IC50 | 2 | — | |
LHQBSXWVTCWYAO
|
6.6 | Kd | 2 | — | |
OJEAHIAKOWKXKB
|
6.6 | IC50 | 2 | — | |
SJBKEBVXIUGVOZ
|
6.6 | IC50 | 2 | — | |
ZDPGILDKHLAGAW
|
6.5 | IC50 | 2 | — | |
RBMAKLWZKDMQGO
|
6.5 | Kd | 2 | — | |
SUOBZGWGYYBNFP
|
6.5 | Kd | 2 | — | |
YZJXMZFIJMZAGN
|
6.5 | IC50 | 2 | — | |
SJGUZBLZMWKMLD
|
6.5 | IC50 | 2 | — | |
IABRAPCYBUUPDG
|
6.5 | Kd | 2 | — | |
MVFXSOJZOSKOQV
|
6.5 | IC50 | 2 | — | |
RYJRIIUWHWEFRG
|
6.5 | IC50 | 2 | — | |
UCPWDZFRWQWHNO
|
6.5 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
6.5 | Kd | 289 | Yes | |
WCJRTXIBTPDRLA
|
6.5 | IC50 | 2 | — | |
BSHJWSAMUHHVFH
|
6.4 | IC50 | 2 | — | |
XEKGZPBWPPGGBY
|
6.4 | IC50 | 2 | — | |
ZLDWNOQHZBTFAQ
|
6.4 | Kd | 2 | — | |
XYQFZKHCIZOACR
|
6.4 | IC50 | 2 | — | |
NGMZJXBTHSWCRY
|
6.4 | IC50 | 2 | — | |
SLUHGHSRHXJQKB
|
6.4 | IC50 | 2 | — | |
SJZKCGAAKXNPOE
|
6.4 | IC50 | 2 | — | |
JYFSQCALHCOVHI
|
6.3 | Kd | 2 | — | |
UHEFRVBGJORHNV
|
6.3 | Kd | 4 | — | |
XJGGJMMBSMTAMQ
|
6.3 | IC50 | 2 | — | |
VXERQKDPAMQZBK
|
6.3 | IC50 | 2 | — | |
UBPYILGKFZZVDX
|
6.3 | Kd | 130 | Yes | |
VOMOOSIWNGQCMM
|
6.3 | IC50 | 2 | — | |
YKNSJONAIIIFGL
|
6.3 | IC50 | 2 | — | |
WZFWHOVNHFFCHJ
|
6.3 | IC50 | 2 | — |