Target Details
| UniProt AC | O43283 |
|---|---|
| Gene Symbol | MAP3K13 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 13 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 234
- Clinical molecules 8
- Avg pChEMBL 7.04
KEGG Pathways (1)
Active Molecules (234)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DHLYOTOZLPRAGO
|
7.1 | IC50 | 2 | — | |
MRVYACMOTKQXLB
|
7.1 | Kd | 2 | — | |
ZIHPELQWBDDGLM
|
7.1 | IC50 | 2 | — | |
ANXJEWGRRMFNLA
|
7.0 | IC50 | 2 | — | |
IZPJZCDJINIEGG
|
7.0 | IC50 | 2 | — | |
VPPAJOKWOOFNML
|
7.0 | Kd | 2 | — | |
WEFXAEVNJQWAFZ
|
7.0 | IC50 | 2 | — | |
JFHNIKLXMSAJQB
|
7.0 | Kd | 2 | — | |
WINHZLLDWRZWRT
|
7.0 | Kd | 201 | Yes | |
CAGRBVWCHLFWPB
|
7.0 | IC50 | 2 | — | |
MVIPEADYCBLILL
|
7.0 | IC50 | 2 | — | |
ZDPGILDKHLAGAW
|
7.0 | IC50 | 2 | — | |
FJLSWQDGOKVNCC
|
7.0 | IC50 | 2 | — | |
GHIXTFPOEFABSP
|
7.0 | IC50 | 2 | — | |
IHMMZBVEKVDJAY
|
7.0 | IC50 | 2 | — | |
ITAHIXXTUMBFLW
|
7.0 | Kd | 2 | — | |
KGGZQEBEACATEW
|
7.0 | IC50 | 2 | — | |
OGENZOBXYZHFIE
|
7.0 | IC50 | 2 | — | |
PWQYILBUZALMLM
|
7.0 | IC50 | 2 | — | |
JVFCJFCGSFJFTE
|
6.9 | IC50 | 2 | — | |
IRPVABHDSJVBNZ
|
6.9 | Kd | 6 | — | |
JWQRMPHYEMLUIF
|
6.9 | IC50 | 2 | — | |
LOGWNXFRIGDZFS
|
6.9 | IC50 | 2 | — | |
MXPDYFZPYGNIET
|
6.9 | IC50 | 2 | — | |
PYILNPDKSAJCQB
|
6.9 | IC50 | 2 | — | |
UQGIRTPAHIWAPS
|
6.9 | IC50 | 2 | — | |
KIKARFDGXOXYJV
|
6.9 | IC50 | 2 | — | |
KRFONFQVWHHIJW
|
6.9 | IC50 | 2 | — | |
GVOOHMLKDGUNOS
|
6.9 | IC50 | 2 | — | |
LXBOBNTVWFNSKG
|
6.9 | IC50 | 2 | — | |
NQPFJBUWMWSZEP
|
6.9 | IC50 | 2 | — | |
YATBHTSLZJEHHE
|
6.9 | IC50 | 2 | — | |
CVXUUYBGGGMSMG
|
6.8 | IC50 | 2 | — | |
KRFONFQVWHHIJW
|
6.8 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
6.8 | Kd | 165 | Yes | |
YRVXIYRJTSIZFV
|
6.8 | IC50 | 2 | — | |
QUJWSXIGZUDUAB
|
6.8 | IC50 | 2 | — | |
HBBBYGQTCMRVDY
|
6.8 | IC50 | 2 | — | |
QIMPNQQBPCORHH
|
6.8 | Kd | 2 | — | |
UOJUEEWSZVRYPU
|
6.8 | Kd | 2 | — | |
WBWAOSSZEUARHN
|
6.8 | IC50 | 2 | — | |
ZTGRUCFMCWRTRS
|
6.8 | Kd | 2 | — | |
BEKZKKDPYXOBQB
|
6.8 | IC50 | 2 | — | |
GGGAYUOZJUDSOF
|
6.8 | Kd | 2 | — | |
RGFWFVVJJAZCNI
|
6.8 | IC50 | 2 | — | |
KERXFSQPGMZQLO
|
6.8 | Kd | 2 | — | |
PIQCTGMSNWUMAF
|
6.8 | Kd | 137 | Yes | |
VSINMMHZZYYOMO
|
6.8 | IC50 | 2 | — | |
GCIKSSRWRFVXBI
|
6.7 | Kd | 109 | Yes | |
LFQVEVGRNHSUDT
|
6.7 | Kd | 2 | — |