Target Details
| UniProt AC | O43283 |
|---|---|
| Gene Symbol | MAP3K13 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 13 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 234
- Clinical molecules 8
- Avg pChEMBL 7.04
KEGG Pathways (1)
Active Molecules (234)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YGSNUGAPYIPPAS
|
7.5 | IC50 | 2 | — | |
GSZNVEWIZSZNJT
|
7.5 | IC50 | 2 | — | |
JHEOSCUBGAKVIR
|
7.5 | IC50 | 2 | — | |
HYQKUJQMGQLFRV
|
7.5 | IC50 | 2 | — | |
CQPIBQJUQSJKOA
|
7.5 | IC50 | 2 | — | |
ITGNDUAJIYAXBQ
|
7.4 | IC50 | 2 | — | |
OEWNOSRZQLNNAS
|
7.4 | IC50 | 2 | — | |
AVWDJSXSWJBVBP
|
7.4 | IC50 | 2 | — | |
FEKFTSSUPZWZPR
|
7.4 | IC50 | 2 | — | |
DZHMDNGHNHTXRV
|
7.4 | IC50 | 2 | — | |
FSTMHVBLNXUGCA
|
7.4 | IC50 | 2 | — | |
GQFXNVBXLWDSDI
|
7.4 | IC50 | 2 | — | |
CSOUOHXVYQKYSZ
|
7.4 | IC50 | 2 | — | |
IVHUDQXUQSQZTQ
|
7.4 | IC50 | 2 | — | |
XZJAQIDXESVVQD
|
7.4 | IC50 | 2 | — | |
WQQYNNJZQBRUAR
|
7.4 | IC50 | 2 | — | |
AVWDJSXSWJBVBP
|
7.3 | IC50 | 2 | — | |
KBBJVNCJPHHXME
|
7.3 | IC50 | 2 | — | |
KKUSYUDWKBDVHV
|
7.3 | IC50 | 2 | — | |
XJJKZADWAKMOHI
|
7.3 | Kd | 2 | — | |
XYWGNKCGTAROOP
|
7.3 | IC50 | 2 | — | |
QKXUHAJFEUPYSC
|
7.3 | Kd | 2 | — | |
QQWVKTNSZANSFF
|
7.3 | IC50 | 2 | — | |
VMLPMFIVJNUHLS
|
7.3 | Kd | 2 | — | |
AMZFWYHDYYBHMD
|
7.3 | IC50 | 2 | — | |
SBJFXIVTSPDBLG
|
7.3 | IC50 | 2 | — | |
ZQBGYFILGRMBEE
|
7.3 | Kd | 2 | — | |
MBVVLBMYGYYEIQ
|
7.3 | IC50 | 2 | — | |
HOAYYWJFTLNUDU
|
7.3 | IC50 | 2 | — | |
PYPUYISPPZTBSN
|
7.2 | IC50 | 2 | — | |
QQWUGDVOUVUTOY
|
7.2 | Kd | 231 | Yes | |
QDLSPDFEDDYQTM
|
7.2 | IC50 | 2 | — | |
FSNRHEHUJCWRAQ
|
7.2 | IC50 | 2 | — | |
NFNPYHGMNVWRTI
|
7.2 | IC50 | 2 | — | |
PSIXMGGMXGEICZ
|
7.2 | IC50 | 2 | — | |
LNSNBRIQENASGL
|
7.2 | Kd | 2 | — | |
IFYGIDLAXXOLQM
|
7.2 | IC50 | 2 | — | |
VDSHJZQIRDEOOY
|
7.2 | Kd | 2 | — | |
IIECRPYGEQYFHR
|
7.2 | IC50 | 2 | — | |
PCPSRYQJUUUZDP
|
7.2 | IC50 | 2 | — | |
GIRIQGHXPJDILQ
|
7.1 | IC50 | 2 | — | |
OGENZOBXYZHFIE
|
7.1 | IC50 | 2 | — | |
RIPVLVJVLRJRKH
|
7.1 | Kd | 2 | — | |
FYFUBZYNKUIYBM
|
7.1 | IC50 | 2 | — | |
UOWUCCPLVGOHMV
|
7.1 | IC50 | 2 | — | |
WMKWBCPSWSWXNF
|
7.1 | IC50 | 2 | — | |
QKAIOVAEPJURBO
|
7.1 | Kd | 2 | — | |
UBLKRXUKBOBBHK
|
7.1 | IC50 | 2 | — | |
HHMAVLGGLJAODV
|
7.1 | IC50 | 2 | — | |
DMZWCKPQTKYLBB
|
7.1 | IC50 | 2 | — |