Target Details
| UniProt AC | O43242 |
|---|---|
| Gene Symbol | PSMD3 |
| Protein Name | 26S proteasome non-ATPase regulatory subunit 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01399 (PCI) PF08375 (Rpn3_C) PF25573 (TPR_PSMD3_N) |
Summary
- Multi-target molecules 29
- Clinical molecules 0
- Avg pChEMBL 7.22
KEGG Pathways (9)
Active Molecules (29)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YUZQDEBWPUFQAF
|
8.2 | IC50 | 38 | — | |
GXJABQQUPOEUTA
|
8.2 | IC50 | 47 | — | |
ORVAWBPOXQNNOV
|
8.1 | IC50 | 38 | — | |
BLMPQMFVWMYDKT
|
8.1 | IC50 | 43 | — | |
PKEANJOUYSERAO
|
7.9 | IC50 | 38 | — | |
MWKSRKSEWLRPBL
|
7.7 | Kd | 1075 | — | |
OGQMVFMKRZZEEH
|
7.7 | IC50 | 38 | — | |
RSKYRPMOCHYBBE
|
7.7 | IC50 | 38 | — | |
CFHYMTUYGRCJAV
|
7.7 | IC50 | 38 | — | |
VMVVXXUNBWJIIZ
|
7.7 | IC50 | 38 | — | |
GAOQGHGKECEBBK
|
7.6 | IC50 | 38 | — | |
ODIWGDQSSAWSIL
|
7.5 | IC50 | 38 | — | |
SODXRIYSSYNQGD
|
7.5 | IC50 | 38 | — | |
VMNWBKJOXQEROK
|
7.5 | IC50 | 38 | — | |
QHQFEEVMNRBZGH
|
7.4 | IC50 | 38 | — | |
VIWWVEXEYFBYDR
|
7.4 | IC50 | 38 | — | |
BBHXTNUZGBPZBK
|
7.1 | IC50 | 38 | — | |
ROTBJYKPNLYFIC
|
7.0 | IC50 | 38 | — | |
PJAVIPGUMNKCGD
|
6.8 | IC50 | 38 | — | |
WMIQZSQGFJUCSD
|
6.8 | IC50 | 38 | — | |
ROTBJYKPNLYFIC
|
6.7 | IC50 | 38 | — | |
WMIQZSQGFJUCSD
|
6.7 | IC50 | 38 | — | |
MSGIVAIQQQASIZ
|
6.5 | IC50 | 38 | — | |
SIBLATFBYYEOCX
|
6.5 | IC50 | 38 | — | |
QYNRQLHUHRJMQN
|
6.4 | IC50 | 38 | — | |
APIXJCOUKQIWCG
|
6.4 | IC50 | 38 | — | |
BLDYDLQKVSQQJZ
|
6.4 | IC50 | 38 | — | |
MCUVOSVWMGVEPT
|
6.2 | IC50 | 38 | — | |
BZRRKMMUABZGLP
|
6.0 | IC50 | 38 | — |