Target Details
| UniProt AC | O30463 |
|---|---|
| Gene Symbol | folA |
| Protein Name | Dihydrofolate reductase |
| Organism | Mycobacterium avium |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00186 (DHFR_1) |
Summary
- Multi-target molecules 146
- Clinical molecules 1
- Avg pChEMBL 8.39
Active Molecules (146)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KZSFROFZPJXGFV
|
8.1 | IC50 | 2 | — | |
DSEIBQNRLLYRRC
|
8.1 | IC50 | 2 | — | |
MXQNQGPRVZDOOS
|
8.0 | IC50 | 2 | — | |
FEZGMOSKDRYDFY
|
8.0 | IC50 | 3 | Yes | |
FGBRLIYQKRWOSO
|
7.9 | IC50 | 2 | — | |
NXCCIJQEAKMFGW
|
7.9 | IC50 | 3 | — | |
KRNZWFKAPBBIRZ
|
7.9 | IC50 | 2 | — | |
LAQLUYMJSYVNIA
|
7.8 | IC50 | 2 | — | |
LJRZTUYWOPFKKK
|
7.8 | IC50 | 2 | — | |
MNHWODGSAAWVCT
|
7.8 | IC50 | 3 | — | |
YVRSSTXQDABQOK
|
7.8 | IC50 | 2 | — | |
KOMMMDLJBSKWOZ
|
7.8 | IC50 | 2 | — | |
MVAHXGRJXVISJS
|
7.8 | IC50 | 2 | — | |
VMBSXLVZCRYQJX
|
7.8 | IC50 | 2 | — | |
HRSHKKZSYXXUHX
|
7.7 | IC50 | 3 | — | |
CHMGVFAMEMAJSZ
|
7.6 | IC50 | 2 | — | |
LUBRVLUNYNBWGR
|
7.6 | IC50 | 2 | — | |
RSQUIUVSFKAGNM
|
7.6 | IC50 | 3 | — | |
VMOVOUMHZIMENS
|
7.5 | IC50 | 2 | — | |
XROWQZMGTMLPOY
|
7.5 | IC50 | 2 | — | |
SXJCFBANUYLDDS
|
7.5 | IC50 | 2 | — | |
OFMQCOABEHAXGV
|
7.4 | IC50 | 3 | — | |
CIUYZEMTWPMSNU
|
7.4 | IC50 | 2 | — | |
VRAFZGTXFNQHGJ
|
7.3 | IC50 | 3 | — | |
QSXKRKHRVCAWRP
|
7.2 | IC50 | 2 | — | |
LQSJMSFERWVWGU
|
7.2 | IC50 | 2 | — | |
LBAODZYBBOYEOK
|
7.1 | IC50 | 3 | — | |
PFSOPZHDFBSZSZ
|
7.0 | IC50 | 3 | — | |
IFIQXNYLZYPKJD
|
7.0 | IC50 | 2 | — | |
KOQCZRWUQXZQNK
|
7.0 | IC50 | 2 | — | |
MJJOMTPSVQORHF
|
7.0 | IC50 | 2 | — | |
QNAXVTNLXFHEBW
|
7.0 | IC50 | 2 | — | |
JQUDVRQNCIBTMP
|
6.9 | IC50 | 3 | — | |
XSIRJSGFRAEBEG
|
6.9 | IC50 | 2 | — | |
GWFSIQAFBODUBN
|
6.8 | IC50 | 2 | — | |
IHHWPKHCZVGDIM
|
6.8 | IC50 | 3 | — | |
CHCXLVNXKKMMBE
|
6.7 | IC50 | 2 | — | |
GKDWTPXQNDNXFE
|
6.5 | IC50 | 2 | — | |
WRYKYFPFYKSJNN
|
6.5 | IC50 | 2 | — | |
YVCCSPPDNARUOV
|
6.5 | IC50 | 3 | — | |
XNDJQQURWLDHAI
|
6.5 | IC50 | 2 | — | |
DINWCFBBTDJSMT
|
6.4 | IC50 | 2 | — | |
MEEJAHCUJQZESD
|
6.2 | IC50 | 2 | — | |
JTNVPKPCMWNPBJ
|
6.2 | IC50 | 2 | — | |
FHGCNTCLPBNZQO
|
6.2 | IC50 | 3 | — | |
HYATWDPIRHVVDH
|
6.2 | IC50 | 3 | — |