Target Details
| UniProt AC | O15530 |
|---|---|
| Gene Symbol | PDPK1 |
| Protein Name | 3-phosphoinositide-dependent protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14593 (PH_3) PF00069 (Pkinase) |
Summary
- Multi-target molecules 228
- Clinical molecules 49
- Avg pChEMBL 7.12
KEGG Pathways (27)
- AMPK signaling pathway
- Aldosterone-regulated sodium reabsorption
- Apoptosis
- Autophagy - animal
- Axon guidance
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Endometrial cancer
- Fc epsilon RI signaling pathway
- Focal adhesion
- FoxO signaling pathway
- IgSF CAM signaling
- Insulin resistance
- Insulin signaling pathway
- Lipid and atherosclerosis
- Neurotrophin signaling pathway
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- PPAR signaling pathway
- Platinum drug resistance
- Prostate cancer
- Proteoglycans in cancer
- Sphingolipid signaling pathway
- T cell receptor signaling pathway
- Thyroid hormone signaling pathway
- Toxoplasmosis
- mTOR signaling pathway
Active Molecules (228)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GHPFSYCYZJKVDZ
|
6.1 | Ki | 18 | Yes | |
NNNVEAQZJOPFCS
|
6.1 | IC50 | 2 | — | |
AWDORCFLUJZUQS
|
6.1 | Ki | 22 | — | |
DFMCXVONDDGQIY
|
6.1 | Ki | 66 | — | |
HHFBDROWDBDFBR
|
6.1 | Ki | 40 | Yes | |
HSYMQQVYGPNCFR
|
6.1 | IC50 | 2 | — | |
PTVPBWWDGZSEAF
|
6.1 | Ki | 63 | — | |
RTDSHUGNRVXRHN
|
6.1 | Ki | 51 | — | |
UGEJLCNSVIVALC
|
6.1 | Ki | 41 | — | |
ULHGAQSVFPOUDY
|
6.1 | Ki | 43 | — | |
VJBYQFPMEPNNCU
|
6.1 | IC50 | 2 | — | |
VKBFHTIUXUCYRQ
|
6.1 | Ki | 66 | — | |
WPHKIQPVPYJNAX
|
6.1 | Ki | 81 | — | |
XJSFDMGICAWQFS
|
6.1 | Ki | 60 | — | |
HHSVICUMCOBRPT
|
6.0 | Ki | 33 | — | |
HVNQYDHDQBJAAH
|
6.0 | IC50 | 3 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MZDKLVOWGIOKTN
|
6.0 | Ki | 80 | — | |
PIQCTGMSNWUMAF
|
6.0 | Ki | 137 | Yes | |
SFPWNTQWFFNJIH
|
6.0 | Ki | 48 | — | |
UQHKJRCFSLMWIA
|
6.0 | IC50 | 3 | — | |
WINHZLLDWRZWRT
|
6.0 | Ki | 66 | — | |
XHORJSJFHVABEA
|
6.0 | Ki | 49 | — | |
ZDNTZQGZVGAPGQ
|
6.0 | IC50 | 4 | — | |
ZGZVRPRSFXRGCF
|
6.0 | Ki | 76 | — | |
ZVWRFVCNQOECJS
|
6.0 | Ki | 71 | — |