Target Details
| UniProt AC | O15530 |
|---|---|
| Gene Symbol | PDPK1 |
| Protein Name | 3-phosphoinositide-dependent protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14593 (PH_3) PF00069 (Pkinase) |
Summary
- Multi-target molecules 228
- Clinical molecules 49
- Avg pChEMBL 7.12
KEGG Pathways (27)
- AMPK signaling pathway
- Aldosterone-regulated sodium reabsorption
- Apoptosis
- Autophagy - animal
- Axon guidance
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Endometrial cancer
- Fc epsilon RI signaling pathway
- Focal adhesion
- FoxO signaling pathway
- IgSF CAM signaling
- Insulin resistance
- Insulin signaling pathway
- Lipid and atherosclerosis
- Neurotrophin signaling pathway
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- PPAR signaling pathway
- Platinum drug resistance
- Prostate cancer
- Proteoglycans in cancer
- Sphingolipid signaling pathway
- T cell receptor signaling pathway
- Thyroid hormone signaling pathway
- Toxoplasmosis
- mTOR signaling pathway
Active Molecules (228)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AOBLBPWPSKBHSI
|
6.6 | Ki | 55 | — | |
GQLWKGVBOIYMTN
|
6.6 | Ki | 35 | — | |
GWJHMRBQEUHFOC
|
6.6 | Ki | 42 | — | |
JCFJQIHDZHHMQT
|
6.6 | Ki | 42 | — | |
QEYGVZZLTIWTEZ
|
6.6 | IC50 | 3 | Yes | |
QPORZABOFXPRHM
|
6.6 | Ki | 18 | — | |
QQWUGDVOUVUTOY
|
6.6 | Ki | 231 | Yes | |
UDFDIIVNIYWXDM
|
6.6 | Ki | 74 | — | |
VBJULRMRDQBSIN
|
6.6 | IC50 | 3 | Yes | |
AAUBJZPZEKVWOC
|
6.6 | IC50 | 3 | — | |
JTGMDPHLGBACAV
|
6.6 | IC50 | 5 | Yes | |
JOAWBRMGMMCJGS
|
6.5 | IC50 | 4 | Yes | |
ORRHVRJUSPCILV
|
6.5 | Ki | 16 | — | |
WVFWTUJEHMVUBG
|
6.5 | Ki | 25 | — | |
XPHWIERLJBFPFV
|
6.5 | Ki | 69 | — | |
ZCCJKVBTHCOISJ
|
6.5 | Ki | 46 | — | |
PPMVOOTZFOABKA
|
6.5 | IC50 | 2 | — | |
TXXYVBLFLGPQOR
|
6.5 | IC50 | 5 | Yes | |
NGFGTMFVWSDFPS
|
6.5 | IC50 | 32 | — | |
SCHFNRDBLZXSFE
|
6.5 | IC50 | 5 | — | |
SRZVWXWGGCOYCF
|
6.5 | IC50 | 2 | — | |
UOSAIBFGDGMQLI
|
6.4 | IC50 | 2 | — | |
QVWIVWPIJUYRRF
|
6.4 | IC50 | 8 | Yes | |
IADKHXRZAFUCSV
|
6.4 | IC50 | 6 | Yes | |
YIGOVOVHNMDCGU
|
6.4 | IC50 | 3 | — | |
AIQDZMUPVYDVLB
|
6.4 | Ki | 48 | — | |
KKYPRNBBPBRJQX
|
6.4 | Ki | 40 | — | |
YEHCNYAQEBQCCS
|
6.4 | Ki | 74 | — | |
XCPMMIISBZJPHR
|
6.4 | IC50 | 3 | — | |
GYPHGCGOSZJXOT
|
6.3 | IC50 | 5 | — | |
FUMCKNCUEAQHCV
|
6.3 | Ki | 103 | — | |
XOOAAYRIVATZNM
|
6.3 | Ki | 55 | — | |
ZWVZORIKUNOTCS
|
6.3 | Ki | 69 | — | |
UZBXYZGLFPRZBL
|
6.3 | IC50 | 2 | — | |
ASDFZNDXNNEZEE
|
6.3 | IC50 | 2 | — | |
SEZFNTZQMWJIAI
|
6.3 | IC50 | 9 | Yes | |
MJSXSLBYCSPRHR
|
6.2 | IC50 | 10 | Yes | |
URECOWLJWSLQCN
|
6.2 | IC50 | 2 | — | |
ZYTRQJFBKVMEAK
|
6.2 | IC50 | 2 | — | |
IKTUPTJGSQCHKN
|
6.2 | IC50 | 2 | — | |
CFIBXVQLBVNOHW
|
6.2 | Ki | 64 | — | |
DWTNLZZEPSCAIH
|
6.2 | Ki | 25 | — | |
GAMJJHMLLXIWRZ
|
6.2 | IC50 | 3 | Yes | |
KRIUNPBAQZGFQA
|
6.2 | Ki | 76 | — | |
NHFDRBXTEDBWCZ
|
6.2 | Ki | 41 | — | |
PCQMERRARZKTPW
|
6.2 | Ki | 68 | — | |
RIBBPSYZBQQTQC
|
6.2 | Ki | 15 | — | |
VKWVIEBXAPQKKA
|
6.2 | Ki | 8 | — | |
YYLKKYCXAOBSRM
|
6.2 | Kd | 191 | — | |
ZCBUQCWBWNUWSU
|
6.2 | IC50 | 59 | — |