Target Details
| UniProt AC | O15393 |
|---|---|
| Gene Symbol | TMPRSS2 |
| Protein Name | Transmembrane protease serine 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF15494 (SRCR_2) PF00089 (Trypsin) |
Summary
- Multi-target molecules 37
- Clinical molecules 0
- Avg pChEMBL 8.06
KEGG Pathways (4)
Active Molecules (37)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MQQNFDZXWVTQEH
|
9.2 | IC50 | 11 | — | |
ZLCINVZAICQINL
|
9.1 | Ki | 4 | — | |
ZLIIZOMJAUACIT
|
9.0 | IC50 | 4 | — | |
YLFDUDAILBTVGN
|
9.0 | Ki | 4 | — | |
NEQGCINBAXAQKD
|
8.9 | IC50 | 5 | — | |
PLLBBBICXMICNE
|
8.9 | IC50 | 4 | — | |
JWFKMTSCIZNZAE
|
8.8 | IC50 | 2 | — | |
JTHVOFMYRRNGPA
|
8.7 | IC50 | 3 | — | |
LNIRCTXHOVOSQG
|
8.6 | IC50 | 3 | — | |
CGFVMUUUSDIEAE
|
8.5 | Ki | 3 | — | |
HJGBKSHYCKEJGU
|
8.5 | Ki | 4 | — | |
VBGVWKFAVGGQCH
|
8.5 | Ki | 4 | — | |
VXMYQVUXZGHVKU
|
8.5 | Ki | 4 | — | |
YXFPBFNFMATBRQ
|
8.5 | IC50 | 4 | — | |
AIAPZNJOJFJSQR
|
8.4 | IC50 | 4 | — | |
WWUOOSJKTRFWDJ
|
8.4 | IC50 | 3 | — | |
DQKGGUJIFZQGEB
|
8.4 | IC50 | 3 | — | |
KQASAMHEMLKUIM
|
8.4 | IC50 | 2 | — | |
HENHNGFKMLDXRP
|
8.3 | IC50 | 3 | — | |
XASIMHXSUQUHLV
|
8.1 | IC50 | 7 | — | |
ZTZVSJUJOHEBFJ
|
8.0 | IC50 | 4 | — | |
GBWLZSRRLJETHI
|
8.0 | IC50 | 5 | — | |
CMECINVDWRULPU
|
7.8 | IC50 | 3 | — | |
NNOFPIZGQIFDSZ
|
7.8 | IC50 | 3 | — | |
WQDFAUJSOUQVHN
|
7.8 | IC50 | 3 | — | |
AIAPZNJOJFJSQR
|
7.8 | IC50 | 4 | — | |
RJBLHAMXODQZMM
|
7.8 | IC50 | 4 | — | |
QKFCYPKTTJCUSZ
|
7.7 | Ki | 8 | — | |
PIYDBRKFQAMHCU
|
7.7 | IC50 | 3 | — | |
DBLNNDOSJLJNTF
|
7.3 | Ki | 4 | — | |
HTOGBQJUJBBWIE
|
7.3 | Ki | 4 | — | |
MISMYWWUBAHTJK
|
7.2 | Ki | 4 | — | |
PXVSKSKOTDZVPH
|
7.2 | Ki | 4 | — | |
XTKGXPFBKPYFDW
|
7.2 | IC50 | 2 | — | |
YKGYIDJEEQRWQH
|
6.9 | IC50 | 6 | — | |
PFGVNLZDWRZPJW
|
6.2 | IC50 | 3 | — | |
OJGDCBLYJGHCIH
|
6.1 | IC50 | 3 | — |