Target Details
| UniProt AC | O15379 |
|---|---|
| Gene Symbol | HDAC3 |
| Protein Name | Histone deacetylase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00850 (Hist_deacetyl) |
Summary
- Multi-target molecules 3,604
- Clinical molecules 474
- Avg pChEMBL 7.22
KEGG Pathways (4)
Active Molecules (3,604)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HYMIWVFCNPTYGW
|
8.9 | IC50 | 4 | — | |
JBBXRYGSCZALTN
|
8.9 | IC50 | 3 | — | |
JBHVIGYZHVIDRH
|
8.9 | IC50 | 3 | — | |
LFXDFXFTOFPLSX
|
8.9 | IC50 | 3 | — | |
LISXISRRNAENFL
|
8.9 | IC50 | 6 | — | |
MRIGHUMOWXZEEI
|
8.9 | IC50 | 4 | — | |
OTDRPXYPNVACGD
|
8.9 | IC50 | 3 | — | |
PJNFGPBZRCJQFS
|
8.9 | IC50 | 12 | Yes | |
WGUXKEANCBSTED
|
8.9 | IC50 | 4 | — | |
YOMPODNRDSCHHL
|
8.9 | IC50 | 4 | — | |
ZFKQNXYKJYAXGV
|
8.9 | IC50 | 3 | — | |
DWVKBTKYJSXCGE
|
8.8 | IC50 | 5 | — | |
FATABLVXWFWXHK
|
8.8 | IC50 | 12 | Yes | |
FQWUNUXAOHTLLG
|
8.8 | Ki | 12 | Yes | |
JAKZKOACZFIOQD
|
8.8 | IC50 | 5 | — | |
JGFQDIKIRZUDAM
|
8.8 | IC50 | 5 | — | |
JIUXQGFMZKHYME
|
8.8 | IC50 | 3 | — | |
KMKZXUFHLBKPAD
|
8.8 | IC50 | 3 | — | |
MTLNSYXCKHAERE
|
8.8 | IC50 | 4 | — | |
NURIFHRHUHZHLY
|
8.8 | IC50 | 4 | Yes | |
WODPQZOZWZAOTM
|
8.8 | IC50 | 4 | — | |
QEQWSYQESDBZGK
|
8.8 | IC50 | 3 | — | |
BLLDUBJDTNVBCR
|
8.8 | IC50 | 3 | — | |
BYAANVBHAFTZAR
|
8.8 | IC50 | 3 | — | |
COFRXQKQVIQIKI
|
8.8 | IC50 | 5 | — | |
CUHDSDLVRCISIT
|
8.8 | IC50 | 11 | — | |
CXXOKIIPISPSNK
|
8.8 | IC50 | 4 | — | |
FCLUGRXEQZESDV
|
8.8 | IC50 | 3 | — | |
FUYHIHBRJCIVJT
|
8.8 | IC50 | 4 | — | |
GWONSPZVVAHEQZ
|
8.8 | IC50 | 4 | — | |
HHIRKUWNXWZRBC
|
8.8 | IC50 | 3 | — | |
IIEGMONUBZNLRW
|
8.8 | IC50 | 5 | — | |
IMRRVABDEDKYSP
|
8.8 | IC50 | 4 | — | |
KBVMOQFPXPZERR
|
8.8 | IC50 | 3 | — | |
KUJIXYVAAZCGKK
|
8.8 | IC50 | 4 | — | |
LTLBNMHJJRQTKA
|
8.8 | IC50 | 4 | — | |
LWUBIRPHWCHAFE
|
8.8 | IC50 | 3 | — | |
MPDRGAGDIRWIMF
|
8.8 | IC50 | 4 | — | |
MYRMVIINVZTODT
|
8.8 | IC50 | 4 | — | |
NKOAGBYPCCDVOF
|
8.8 | IC50 | 4 | — | |
OCEYRAXLYFYSEZ
|
8.8 | IC50 | 3 | — | |
PGTVKKLHFBLXOX
|
8.8 | IC50 | 4 | — | |
PKQXIFMKLJMAQQ
|
8.8 | IC50 | 4 | — | |
PVFXNOGMVQSUGR
|
8.8 | IC50 | 4 | — | |
QBWTZABUPQHVIG
|
8.8 | IC50 | 4 | — | |
QZALBIBLDLTXIY
|
8.8 | IC50 | 4 | — | |
RIHKXPFNMAZMOA
|
8.8 | IC50 | 11 | — | |
SPZAYRRDKQWOGT
|
8.8 | IC50 | 4 | — | |
UATFOQLTQPSSIR
|
8.8 | IC50 | 3 | — | |
WEUZJBFBMQCGSG
|
8.8 | IC50 | 11 | — |