Target Details
| UniProt AC | O15379 |
|---|---|
| Gene Symbol | HDAC3 |
| Protein Name | Histone deacetylase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00850 (Hist_deacetyl) |
Summary
- Multi-target molecules 3,604
- Clinical molecules 474
- Avg pChEMBL 7.22
KEGG Pathways (4)
Active Molecules (3,604)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GREXOPZRGSQSHE
|
9.5 | IC50 | 11 | — | |
VXQMEGLYMWVBHB
|
9.5 | IC50 | 6 | — | |
ZIXGFQGSZCYOCA
|
9.5 | IC50 | 11 | — | |
PLWBVDLCWWJINE
|
9.5 | IC50 | 4 | — | |
KIHNNQQNYQLDGM
|
9.5 | IC50 | 5 | — | |
NLIBKESLXRYMGS
|
9.5 | IC50 | 4 | — | |
YMGFKZMMMPLPMK
|
9.5 | IC50 | 3 | — | |
RCHCXFHRGGHVRF
|
9.4 | IC50 | 3 | — | |
LYACRWFTZJMETD
|
9.4 | IC50 | 4 | — | |
MQRZDKMXNGUVAV
|
9.4 | IC50 | 3 | — | |
VCQGMJZYDYIFCF
|
9.4 | IC50 | 4 | — | |
MYZPAEFNFJXMAN
|
9.4 | IC50 | 3 | — | |
RNOLVRZGDPVERA
|
9.4 | IC50 | 3 | — | |
AEDUBEGTPWKDCX
|
9.4 | IC50 | 6 | — | |
AEDUBEGTPWKDCX
|
9.4 | IC50 | 12 | Yes | |
BPGNCVTVTQPXKS
|
9.4 | IC50 | 3 | — | |
HOFXGVRUBPUUSI
|
9.4 | IC50 | 3 | — | |
JPXOLQFKWRYZSF
|
9.4 | IC50 | 4 | — | |
KPLSOOZZGITXDX
|
9.4 | IC50 | 3 | — | |
MGSMSINQVPOBFG
|
9.4 | IC50 | 12 | — | |
NXFALCZBQFKESM
|
9.4 | IC50 | 14 | Yes | |
UWIASJNPIIGSRX
|
9.4 | IC50 | 4 | — | |
VOCUPJYYWCXUPO
|
9.4 | IC50 | 3 | — | |
XVLFDROZMUKWLL
|
9.4 | IC50 | 4 | — | |
HACPSCZAVPAEID
|
9.4 | IC50 | 4 | — | |
LEGQHRJRAAFESX
|
9.4 | IC50 | 4 | — | |
LHNROLRKNQLRIY
|
9.4 | IC50 | 4 | — | |
XGCLYPPRQZTIBB
|
9.4 | IC50 | 4 | — | |
DDNWDPJEUUPJGI
|
9.3 | IC50 | 3 | — | |
JBCPWLASJZAEQC
|
9.3 | IC50 | 4 | — | |
OOXJXQXMYMAFJQ
|
9.3 | IC50 | 4 | — | |
TUMLTUXMYBNUKT
|
9.3 | IC50 | 4 | — | |
UTPAUKFZOVQYCD
|
9.3 | IC50 | 3 | — | |
PSAATLQEQBLXDQ
|
9.3 | IC50 | 4 | — | |
CIVLRUVGMDDSMH
|
9.3 | IC50 | 4 | — | |
KIGCDQVXODFLML
|
9.3 | IC50 | 5 | — | |
SCGYNYNZVFVIFE
|
9.3 | IC50 | 4 | — | |
VWZPZBCVBMLKHY
|
9.3 | IC50 | 4 | — | |
ZRFLMIZPTHEEJS
|
9.3 | IC50 | 4 | — | |
AZODTJZLKVAKDP
|
9.3 | IC50 | 4 | — | |
CDWXREOLGKHQQP
|
9.3 | IC50 | 3 | — | |
DEPGTCNZKXMKRK
|
9.3 | IC50 | 3 | — | |
SNGOLLQHPCZCCY
|
9.3 | IC50 | 4 | — | |
GSBGMIOHBWZCMF
|
9.3 | IC50 | 3 | — | |
KHFJYYIYUAHKHW
|
9.3 | IC50 | 4 | — | |
MZCMRPRNHRPNAJ
|
9.3 | IC50 | 2 | — | |
NGTLBSGOPOBCFZ
|
9.3 | IC50 | 5 | — | |
BZIQIFZLMIFLBH
|
9.3 | IC50 | 4 | — | |
DOCUUNQBCZHNKR
|
9.3 | IC50 | 4 | — | |
IACGDSJQDVSAPH
|
9.2 | IC50 | 5 | — |