Target Details
| UniProt AC | O15197 |
|---|---|
| Gene Symbol | EPHB6 |
| Protein Name | Ephrin type-B receptor 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF07699 (Ephrin_rec_like) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF07647 (SAM_2) |
Summary
- Multi-target molecules 42
- Clinical molecules 19
- Avg pChEMBL 7.03
Active Molecules (42)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AQSSMEORRLJZLU
|
9.2 | Kd | 34 | Yes | |
SEJGTFPOEJWEGG
|
8.9 | Kd | 149 | — | |
VAARYSWULJUGST
|
8.7 | Kd | 119 | Yes | |
SHPFDGWALWEPGS
|
8.3 | Kd | 35 | — | |
KTEIFNKAUNYNJU
|
8.2 | Kd | 114 | — | |
BEMNJULZEQTDJY
|
8.2 | Kd | 8 | — | |
LOLPPWBBNUVNQZ
|
7.9 | Kd | 97 | Yes | |
ALKJNCZNEOTEMP
|
7.6 | Kd | 55 | — | |
CXQHYVUVSFXTMY
|
7.6 | Kd | 154 | — | |
GCIKSSRWRFVXBI
|
7.5 | Kd | 109 | Yes | |
MPVGZUGXCQEXTM
|
7.5 | Kd | 61 | Yes | |
ZBNZXTGUTAYRHI
|
7.5 | Kd | 102 | Yes | |
YABJJWZLRMPFSI
|
7.4 | Kd | 34 | — | |
QYZOGCMHVIGURT
|
7.3 | Kd | 26 | Yes | |
UHTHHESEBZOYNR
|
7.1 | Kd | 66 | Yes | |
CUIHSIWYWATEQL
|
7.1 | Kd | 61 | Yes | |
UIARLYUEJFELEN
|
7.0 | Kd | 289 | Yes | |
VYPGLYMWNDRFGZ
|
6.9 | Kd | 12 | — | |
YYLKKYCXAOBSRM
|
6.9 | Kd | 191 | — | |
XZXHXSATPCNXJR
|
6.8 | Kd | 165 | Yes | |
XKFTZKGMDDZMJI
|
6.8 | Kd | 64 | Yes | |
HKSZLNNOFSGOKW
|
6.7 | Kd | 408 | — | |
PIQCTGMSNWUMAF
|
6.7 | Kd | 137 | Yes | |
XXJWYDDUDKYVKI
|
6.7 | Kd | 52 | — | |
HXHAJRMTJXHJJZ
|
6.7 | Kd | 52 | Yes | |
ZCCPLJOKGAACRT
|
6.7 | Kd | 599 | — | |
MLDQJTXFUGDVEO
|
6.6 | Kd | 85 | Yes | |
HVXKQKFEHMGHSL
|
6.6 | Kd | 21 | — | |
UQRCJCNVNUFYDX
|
6.6 | Kd | 27 | — | |
JOOXLOJCABQBSG
|
6.5 | Kd | 139 | — | |
NHHQJBCNYHBUSI
|
6.5 | Kd | 220 | — | |
QQWUGDVOUVUTOY
|
6.5 | Kd | 231 | Yes | |
RITAVMQDGBJQJZ
|
6.4 | Kd | 43 | — | |
BFSMGDJOXZAERB
|
6.4 | Kd | 33 | — | |
WKDACQVEJIVHMZ
|
6.3 | Kd | 46 | — | |
HHZIURLSWUIHRB
|
6.3 | Kd | 57 | Yes | |
DKZYXHCYPUVGAF
|
6.3 | Kd | 112 | — | |
NXSJMRCTGYTSTK
|
6.2 | Kd | 200 | — | |
OMZCMEYTWSXEPZ
|
6.2 | Kd | 43 | Yes | |
AUOSKLDNVNGKRR
|
6.2 | Kd | 6 | — | |
YZDJQTHVDDOVHR
|
6.1 | Kd | 23 | — | |
WINHZLLDWRZWRT
|
6.0 | Kd | 201 | Yes |